Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
CD63 antigen (Homo sapiens (Human)) | BDBM212272 ((R)-(4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]p...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 33 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212270 (6-(6-amino-5-methylpyrazin-2-yl)-N-(4-(4-(oxetan-3...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 51 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212271 (6-(6-aminopyrazin-2-yl)-N-(4-(4-(oxetan-3-yl)piper...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | US Patent | n/a | n/a | 80 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM324284 ((R)-1-(tert-butyl)-N-(8-(2-((1-methyl-1H-pyrazol-4...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 82 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of CD63 (unknown origin) assessed as FcepsilonR induced basophil activation | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00926 BindingDB Entry DOI: 10.7270/Q23B641C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212277 (US11517570, Example Kn.-1: | US9290505, 6-(5-amino...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 101 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212274 (2-(5-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]pyrazi...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 120 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212275 (2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 128 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212273 (6-(6-aminopyrazin-2-yl)-5-methyl-N-(4-(4-(oxetan-3...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 157 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212276 (2-(5-((6-(6-amino-5-methylpyrazin-2-yl)imidazo[1,2...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 167 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212279 (US11517570, Example Kn.-3: | US9290505, 6-(5-amino...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 250 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212280 (US11517570, Example Kn.-4: | US9290505, 6-(6-amino...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 734 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CD63 antigen (Homo sapiens (Human)) | BDBM212278 (US11517570, Example Kn.-2: | US9290505, 6-(3-amino...) | MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 809 | n/a | n/a | n/a | n/a | 7.0 | n/a |
Gilead Sciences, Inc. US Patent | Assay Description Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca... | US Patent US9290505 (2016) BindingDB Entry DOI: 10.7270/Q2TB15RT | |||||||||||
More data for this Ligand-Target Pair |