Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
G-protein coupled receptor 39 (Mus musculus) | BDBM50030767 (CHEMBL3342365) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 365 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50232401 (CHEMBL4077818) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ... | J Med Chem 60: 886-898 (2017) Article DOI: 10.1021/acs.jmedchem.6b00648 BindingDB Entry DOI: 10.7270/Q2VT1VBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030769 (CHEMBL3342363) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030770 (CHEMBL3342362) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030771 (CHEMBL3342361) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030772 (CHEMBL3342360) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030773 (CHEMBL3342359) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 115 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030789 (CHEMBL3341764) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030790 (CHEMBL3342357) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030787 (CHEMBL3342366) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030786 (CHEMBL3342367) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030785 (CHEMBL3342368) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 304 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030784 (CHEMBL3342369) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.61E+3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030783 (CHEMBL3342370) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030782 (CHEMBL3342371) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030781 (CHEMBL3342372) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 17 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030780 (CHEMBL3342373) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 34 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030779 (CHEMBL3342374) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030778 (CHEMBL3342375) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 185 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030777 (CHEMBL3342376) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030776 (CHEMBL3342377) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030775 (CHEMBL3342378) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50232367 (CHEMBL4093273) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ... | J Med Chem 60: 886-898 (2017) Article DOI: 10.1021/acs.jmedchem.6b00648 BindingDB Entry DOI: 10.7270/Q2VT1VBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50232401 (CHEMBL4077818) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 180 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ... | J Med Chem 60: 886-898 (2017) Article DOI: 10.1021/acs.jmedchem.6b00648 BindingDB Entry DOI: 10.7270/Q2VT1VBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50232391 (CHEMBL4100119) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ... | J Med Chem 60: 886-898 (2017) Article DOI: 10.1021/acs.jmedchem.6b00648 BindingDB Entry DOI: 10.7270/Q2VT1VBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 39 (Mus musculus) | BDBM50030768 (CHEMBL3342364) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.72E+3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at mouse GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair |