Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM50086441 (CHEMBL3426225 | US10266537, Compound 3) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc. | Assay Description The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot... | Bioorg Med Chem Lett 17: 3562-9 (2007) BindingDB Entry DOI: 10.7270/Q21C2065 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111473 (4-Methyl-N-(4-(2-morpholinoethoxy) phenyl)-3-(4-(p...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111449 (4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 136 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111466 (4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM50237710 (4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 214 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111456 (N-(3-bromo-5-(trifluoromethyl) phenyl)-4-methyl-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 219 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111455 (N-(3,5-bis(trifluoromethyl) phenyl)-4-methyl-3-(4-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 259 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111465 (N-(5-chloropyridin-2-yl)-4-methyl-3-(4-(pyridin-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 305 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111452 (N-(4-bromophenyl)-4-methyl-3-(4-(pyridin-3-yl) pyr...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 483 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111460 (N-(3-acetylphenyl)-4-methyl-3-(4-(pyridin-3-yl) py...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 542 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111453 (N-(2-fluorophenyl)-4-methyl-3-(4-(pyridin-3-yl) py...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 569 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111451 (N-(4-methoxyphenyl)-4-methyl-3-(4-(pyridin-3-yl) p...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 924 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111459 (N-(2, 6-dimethylphenyl)-4-methyl-3-(4-(pyridin-3-y...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 956 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111454 (N-(3-fluorophenyl)-4-methyl-3-(4-(pyridin-3-yl) py...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111457 (4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111450 (N-(3, 4-dichlorophenyl)-4-methyl-3-(4-(pyridin-3-y...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111462 (4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111464 (4-Methyl-N-(pyridin-2-yl)-3-(4-(pyridin-3-yl) pyri...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111467 (4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111463 (4-Methyl-N-(pyridin-3-yl)-3-(4-(pyridin-3-yl) pyri...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111461 (N-(3-methoxyphenyl)-4-methyl-3-(4-(pyridin-3-yl) p...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.24E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111448 (N-(3-chloro-4-fluorophenyl)-4-methyl-3-(4-(pyridin...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111468 (N-(4-(3-(dimethylamino)propoxy) phenyl)-4-methyl- ...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.32E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111469 (N-(4-(2-(dimethylamino)ethoxy)phenyl)-4-methyl-3-(...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111471 (4-Methyl-3-(4-(pyridin-3-yl) pyrimidin-2-ylamino)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111474 (4-Methyl-N-(4-(3-morpholinopropoxy) phenyl)-3-(4-(...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111470 (N-(4-(2-(diethylamino)ethoxy)phenyl)-4-methyl-3-(4...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Breakpoint cluster region protein [1-693] (Homo sapiens (Human)) | BDBM111472 (4-Methyl-N-(4-(2-(piperidin-1-yl) ethoxy) phenyl)-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Xi'an Jiaotong University, No. 76, Yanta West Road, Xi'an, 710061, China | Assay Description ATP (6.021 μM) and substrate (457.7 nM) were used. Kinase, substrate peptide, and inhibitor were added in a 384-well plate. The reaction was s... | Chem Biol Drug Des 83: 592-9 (2014) Article DOI: 10.1111/cbdd.12272 BindingDB Entry DOI: 10.7270/Q2GX497N | |||||||||||
More data for this Ligand-Target Pair |