Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382126 (4-(4-((4'-(1-cyanocyclopropyl)-3,4,5,6-tetrahydro-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382141 (4-(4-((4-fluoro-4'-methyl-3,4,5,6-tetrahydro-[1,1'...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382128 (4-(4-((4'-methoxy-3,4,5,6-tetrahydro-[1,1'-bipheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382129 (4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 275 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382130 (4-(4-((2-(6-amino-5-(trifluoromethyl)pyridin-3-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382131 (4-(4-((2-(5,6,7,8-tetrahydronaphthalen-2-yl)cycloh...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 275 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382132 (4-(4-([1,1'-bi(cyclohexane)]-1,1'-dien-2-ylmethoxy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382133 (4-(4-((2-(6-methoxypyridin-3-yl)cyclohex-1-en-1-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382134 (4-(4-((2-(4-(1-cyanocyclopropyl)phenyl)cyclohept-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 275 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382134 (4-(4-((2-(4-(1-cyanocyclopropyl)phenyl)cyclohept-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382136 (4-(4-((2-(p-tolyl)cyclohept-1-en-1-yl)methoxy)phen...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 275 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382137 (4-(4-((4-(4-(1-cyanocyclopropyl)phenyl)-5,6-dihydr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382138 (4-(4-((4-(5,6,7,8-tetrahydronaphthalen-2-yl)-5,6-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382139 (4-(4-((2-(p-tolyloxy)cyclohex-1-en-1-yl)methoxy)ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382140 (4-(4-((4'-(1-cyanocyclopropyl)-4-methyl-3,4,5,6-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM382127 (4-(4-((2-(4,5,6,7-tetrahydrobenzo[d]thiazol-2-yl)c...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 2.75E+3 | n/a | n/a | n/a | n/a |
IRBM/Merck | Assay Description Beta (β) arrestin 2 Interaction Assay (BRET assay) was performed using CHO-K1 cells stably expressing the GPR120 receptor using β-galactosi... | Bioorg Med Chem Lett 18: 3456-61 (2008) BindingDB Entry DOI: 10.7270/Q2154KBP | |||||||||||
More data for this Ligand-Target Pair |