Found 29 hits Enz. Inhib. hit(s) with all data for entry = 50003545 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50222968
![PNG](/data/jpeg/tenK5022/BindingDB_50222968.png) (Cipralisant | GT-2331)Show InChI InChI=1S/C14H20N2/c1-14(2,3)7-5-4-6-11-8-12(11)13-9-15-10-16-13/h9-12H,5,7-8H2,1-3H3,(H,15,16)/t11-,12-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| 0.126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472544
![PNG](/data/jpeg/tenK5047/BindingDB_50472544.png) (Iodoproxyfan)Show InChI InChI=1S/C13H15IN2O/c14-12-5-3-11(4-6-12)9-17-7-1-2-13-8-15-10-16-13/h3-6,8,10H,1-2,7,9H2,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 0.126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472544
![PNG](/data/jpeg/tenK5047/BindingDB_50472544.png) (Iodoproxyfan)Show InChI InChI=1S/C13H15IN2O/c14-12-5-3-11(4-6-12)9-17-7-1-2-13-8-15-10-16-13/h3-6,8,10H,1-2,7,9H2,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 0.126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472543
![PNG](/data/jpeg/tenK5047/BindingDB_50472543.png) (CHEMBL278276)Show SMILES [H][C@]1(C[C@@]1([H])c1c[nH]cn1)\C=C\[C@@H](N)CC1CCCCC1 Show InChI InChI=1S/C16H25N3/c17-14(8-12-4-2-1-3-5-12)7-6-13-9-15(13)16-10-18-11-19-16/h6-7,10-15H,1-5,8-9,17H2,(H,18,19)/b7-6+/t13-,14-,15-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 0.398 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50214615
![PNG](/data/jpeg/tenK5021/BindingDB_50214615.png) (CHEBI:64177 | Clobenpropit)Show InChI InChI=1S/C14H17ClN4S/c15-12-5-3-11(4-6-12)8-18-14(16)20-7-1-2-13-9-17-10-19-13/h3-6,9-10H,1-2,7-8H2,(H2,16,18)(H,17,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50214615
![PNG](/data/jpeg/tenK5021/BindingDB_50214615.png) (CHEBI:64177 | Clobenpropit)Show InChI InChI=1S/C14H17ClN4S/c15-12-5-3-11(4-6-12)8-18-14(16)20-7-1-2-13-9-17-10-19-13/h3-6,9-10H,1-2,7-8H2,(H2,16,18)(H,17,19) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
KEGG PC cid PC sid UniChem
Similars
| Article PubMed
| 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50050180
![PNG](/data/jpeg/tenK5005/BindingDB_50050180.png) (4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)Show InChI InChI=1S/C13H15BrN2O/c14-12-5-3-11(4-6-12)9-17-7-1-2-13-8-15-10-16-13/h3-6,8,10H,1-2,7,9H2,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 1.26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50050180
![PNG](/data/jpeg/tenK5005/BindingDB_50050180.png) (4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)Show InChI InChI=1S/C13H15BrN2O/c14-12-5-3-11(4-6-12)9-17-7-1-2-13-8-15-10-16-13/h3-6,8,10H,1-2,7,9H2,(H,15,16) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 1.26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50215536
![PNG](/data/jpeg/tenK5021/BindingDB_50215536.png) ((R)-Alpha-Methylhistamine | CHEBI:73337 | CHEMBL26...)Show InChI InChI=1S/C6H11N3/c1-5(7)2-6-3-8-4-9-6/h3-5H,2,7H2,1H3,(H,8,9)/t5-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Similars
| Article PubMed
| 2.51 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472551
![PNG](/data/jpeg/tenK5047/BindingDB_50472551.png) (proxifan | proxyfan)Show InChI InChI=1S/C13H16N2O/c1-2-5-12(6-3-1)10-16-8-4-7-13-9-14-11-15-13/h1-3,5-6,9,11H,4,7-8,10H2,(H,14,15) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
PC cid PC sid UniChem
| Article PubMed
| 3.16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50127607
![PNG](/data/jpeg/tenK5012/BindingDB_50127607.png) ((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)Show InChI InChI=1S/C6H9N3/c7-5-1-4(5)6-2-8-3-9-6/h2-5H,1,7H2,(H,8,9)/t4-,5-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472551
![PNG](/data/jpeg/tenK5047/BindingDB_50472551.png) (proxifan | proxyfan)Show InChI InChI=1S/C13H16N2O/c1-2-5-12(6-3-1)10-16-8-4-7-13-9-14-11-15-13/h1-3,5-6,9,11H,4,7-8,10H2,(H,14,15) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
PC cid PC sid UniChem
| Article PubMed
| 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description PKi was measured by Histamine H3 receptor binding assay (N-alpha-MeHA) on rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472556
![PNG](/data/jpeg/tenK5047/BindingDB_50472556.png) (CHEMBL428343)Show InChI InChI=1S/C13H23N3O/c14-12(6-13-7-15-10-16-13)9-17-8-11-4-2-1-3-5-11/h7,10-12H,1-6,8-9,14H2,(H,15,16)/t12-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 12.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472542
![PNG](/data/jpeg/tenK5047/BindingDB_50472542.png) (CHEMBL18554)Show SMILES [H][C@@]1(C[C@]1([H])c1c[nH]cn1)NC(=O)[C@@H](N)Cc1ccccc1 Show InChI InChI=1S/C15H18N4O/c16-12(6-10-4-2-1-3-5-10)15(20)19-13-7-11(13)14-8-17-9-18-14/h1-5,8-9,11-13H,6-7,16H2,(H,17,18)(H,19,20)/t11-,12-,13-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50127605
![PNG](/data/jpeg/tenK5012/BindingDB_50127605.png) ((1S,2S)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)Show InChI InChI=1S/C6H9N3/c7-5-1-4(5)6-2-8-3-9-6/h2-5H,1,7H2,(H,8,9)/t4-,5-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472547
![PNG](/data/jpeg/tenK5047/BindingDB_50472547.png) (CHEMBL19413)Show InChI InChI=1S/C13H17N3O/c14-12(6-13-7-15-10-16-13)9-17-8-11-4-2-1-3-5-11/h1-5,7,10,12H,6,8-9,14H2,(H,15,16)/t12-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 50.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472545
![PNG](/data/jpeg/tenK5047/BindingDB_50472545.png) (CHEMBL418736)Show InChI InChI=1S/C13H16BrN3O/c14-11-3-1-10(2-4-11)7-18-8-12(15)5-13-6-16-9-17-13/h1-4,6,9,12H,5,7-8,15H2,(H,16,17)/t12-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 79.4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472546
![PNG](/data/jpeg/tenK5047/BindingDB_50472546.png) (CHEMBL19469)Show SMILES [H][C@]1(C[C@@]1([H])c1c[nH]cn1)\C=C/[C@@H](N)CC1CCCCC1 Show InChI InChI=1S/C16H25N3/c17-14(8-12-4-2-1-3-5-12)7-6-13-9-15(13)16-10-18-11-19-16/h6-7,10-15H,1-5,8-9,17H2,(H,18,19)/b7-6-/t13-,14-,15-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472552
![PNG](/data/jpeg/tenK5047/BindingDB_50472552.png) (CHEMBL18696)Show InChI InChI=1S/C14H18N4O/c15-13(8-11-4-2-1-3-5-11)14(19)17-7-6-12-9-16-10-18-12/h1-5,9-10,13H,6-8,15H2,(H,16,18)(H,17,19)/t13-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472559
![PNG](/data/jpeg/tenK5047/BindingDB_50472559.png) ((S)-Alpha-Methylhistamine | CHEMBL11919)Show InChI InChI=1S/C6H11N3/c1-5(7)2-6-3-8-4-9-6/h3-5H,2,7H2,1H3,(H,8,9)/t5-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE PC cid PC sid UniChem
| Article PubMed
| 158 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472560
![PNG](/data/jpeg/tenK5047/BindingDB_50472560.png) (CHEMBL276987)Show InChI InChI=1S/C13H23N3O/c14-12(6-13-7-15-10-16-13)9-17-8-11-4-2-1-3-5-11/h7,10-12H,1-6,8-9,14H2,(H,15,16)/t12-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 158 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472558
![PNG](/data/jpeg/tenK5047/BindingDB_50472558.png) (CHEMBL18685)Show InChI InChI=1S/C13H16BrN3O/c14-11-3-1-10(2-4-11)7-18-8-12(15)5-13-6-16-9-17-13/h1-4,6,9,12H,5,7-8,15H2,(H,16,17)/t12-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 199 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472550
![PNG](/data/jpeg/tenK5047/BindingDB_50472550.png) (CHEMBL19329)Show InChI InChI=1S/C13H16IN3O/c14-11-3-1-10(2-4-11)7-18-8-12(15)5-13-6-16-9-17-13/h1-4,6,9,12H,5,7-8,15H2,(H,16,17)/t12-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 199 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472549
![PNG](/data/jpeg/tenK5047/BindingDB_50472549.png) (CHEBI:16255 | HISTIDINOL)Show InChI InChI=1S/C6H11N3O/c7-5(3-10)1-6-2-8-4-9-6/h2,4-5,10H,1,3,7H2,(H,8,9)/t5-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE KEGG PC cid PC sid UniChem
| Article PubMed
| 251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472557
![PNG](/data/jpeg/tenK5047/BindingDB_50472557.png) (CHEMBL416365)Show InChI InChI=1S/C13H16IN3O/c14-11-3-1-10(2-4-11)7-18-8-12(15)5-13-6-16-9-17-13/h1-4,6,9,12H,5,7-8,15H2,(H,16,17)/t12-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472554
![PNG](/data/jpeg/tenK5047/BindingDB_50472554.png) (CHEMBL280034)Show InChI InChI=1S/C13H17N3O/c14-12(6-13-7-15-10-16-13)9-17-8-11-4-2-1-3-5-11/h1-5,7,10,12H,6,8-9,14H2,(H,15,16)/t12-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 316 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472548
![PNG](/data/jpeg/tenK5047/BindingDB_50472548.png) (CHEMBL418734)Show InChI InChI=1S/C7H13N3O/c1-11-4-6(8)2-7-3-9-5-10-7/h3,5-6H,2,4,8H2,1H3,(H,9,10)/t6-/m0/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| 1.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472553
![PNG](/data/jpeg/tenK5047/BindingDB_50472553.png) (CHEMBL19588)Show InChI InChI=1S/C6H11N3O/c7-5(3-10)1-6-2-8-4-9-6/h2,4-5,10H,1,3,7H2,(H,8,9)/t5-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
PC cid PC sid UniChem
| Article PubMed
| 1.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Affinity for histamine H3 receptor in rat cerebral cortex. |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |
Histamine H3 receptor
(Rattus norvegicus (rat)) | BDBM50472555
![PNG](/data/jpeg/tenK5047/BindingDB_50472555.png) (CHEMBL18884)Show InChI InChI=1S/C14H18N4O/c15-13(8-11-4-2-1-3-5-11)14(19)17-7-6-12-9-16-10-18-12/h1-5,9-10,13H,6-8,15H2,(H,16,18)(H,17,19)/t13-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kuopio
Curated by ChEMBL
| Assay Description Binding affinity of compound against Histamine H3 receptor |
J Med Chem 42: 1193-202 (1999)
Article DOI: 10.1021/jm980408v BindingDB Entry DOI: 10.7270/Q20Z760D |
More data for this Ligand-Target Pair | |