Search and Browse
Download
Enter Data
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Mitogen-activated protein kinase 10 (Homo sapiens (Human)) | BDBM50550131 (CHEMBL4754904) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet  | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK10 using peptide substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 10 (Homo sapiens (Human)) | BDBM50550132 (CHEMBL4749658) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 780 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK10 using peptide substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Glycogen synthase kinase-3 alpha (Homo sapiens (Human)) | BDBM50550131 (CHEMBL4754904) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human GSK3alpha S449A mutant (2 to end residues) using YRRAAVPPSPSLSR peptide as substrate incubated for 40 mins in presenc... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 10 (Homo sapiens (Human)) | BDBM50550129 (CHEMBL4744511) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK10 using peptide substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Glycogen synthase kinase-3 alpha (Homo sapiens (Human)) | BDBM50550132 (CHEMBL4749658) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human GSK3alpha S449A mutant (2 to end residues) using YRRAAVPPSPSLSR peptide as substrate incubated for 40 mins in presenc... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Glycogen synthase kinase-3 alpha (Homo sapiens (Human)) | BDBM50550133 (CHEMBL4754518) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human GSK3alpha S449A mutant (2 to end residues) using YRRAAVPPSPSLSR peptide as substrate incubated for 40 mins in presenc... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 10 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK10 using peptide substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Glycogen synthase kinase-3 alpha (Homo sapiens (Human)) | BDBM50550129 (CHEMBL4744511) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human GSK3alpha S449A mutant (2 to end residues) using YRRAAVPPSPSLSR peptide as substrate incubated for 40 mins in presenc... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550131 (CHEMBL4754904) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 10 (Homo sapiens (Human)) | BDBM50550133 (CHEMBL4754518) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK10 using peptide substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550129 (CHEMBL4744511) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550132 (CHEMBL4749658) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Glycogen synthase kinase-3 alpha (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human GSK3alpha S449A mutant (2 to end residues) using YRRAAVPPSPSLSR peptide as substrate incubated for 40 mins in presenc... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550137 (CHEMBL4750817) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550133 (CHEMBL4754518) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550128 (CHEMBL4777902) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550134 (CHEMBL4748932) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550142 (CHEMBL4799148) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 8 (Homo sapiens (Human)) | BDBM50550132 (CHEMBL4749658) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK8 using ATF2 as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintilla... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 8 (Homo sapiens (Human)) | BDBM50550133 (CHEMBL4754518) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK8 using ATF2 as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintilla... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 8 (Homo sapiens (Human)) | BDBM50550131 (CHEMBL4754904) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK8 using ATF2 as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintilla... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 8 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK8 using ATF2 as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintilla... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 8 (Homo sapiens (Human)) | BDBM50550129 (CHEMBL4744511) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of full length recombinant human MAPK8 using ATF2 as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintilla... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Homeodomain-interacting protein kinase 1 (Homo sapiens (Human)) | BDBM50550133 (CHEMBL4754518) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scinti... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Homeodomain-interacting protein kinase 1 (Homo sapiens (Human)) | BDBM50550132 (CHEMBL4749658) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scinti... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Homeodomain-interacting protein kinase 1 (Homo sapiens (Human)) | BDBM50550131 (CHEMBL4754904) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scinti... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Homeodomain-interacting protein kinase 1 (Homo sapiens (Human)) | BDBM50550129 (CHEMBL4744511) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scinti... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Homeodomain-interacting protein kinase 1 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scinti... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| SNF-related serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50550133 (CHEMBL4754518) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human SNRK E97G/P116A mutant (1 to 505 residues) using KKLRRTLSFAEPG peptide as substrate incubated for 40 mins in presence... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| SNF-related serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50550132 (CHEMBL4749658) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human SNRK E97G/P116A mutant (1 to 505 residues) using KKLRRTLSFAEPG peptide as substrate incubated for 40 mins in presence... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| SNF-related serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50550131 (CHEMBL4754904) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human SNRK E97G/P116A mutant (1 to 505 residues) using KKLRRTLSFAEPG peptide as substrate incubated for 40 mins in presence... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| SNF-related serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50550129 (CHEMBL4744511) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human SNRK E97G/P116A mutant (1 to 505 residues) using KKLRRTLSFAEPG peptide as substrate incubated for 40 mins in presence... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| SNF-related serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human SNRK E97G/P116A mutant (1 to 505 residues) using KKLRRTLSFAEPG peptide as substrate incubated for 40 mins in presence... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550130 (CHEMBL4785960) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.34E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550138 (CHEMBL4749115) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.45E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.46E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550139 (CHEMBL4786052) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550136 (CHEMBL4765173) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550135 (CHEMBL4794407) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550141 (CHEMBL4791951) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550140 (CHEMBL4745254) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Displacement of tracer K5 from N-terminal nanoluciferase-tagged RIOK2 (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET ass... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Serine/threonine-protein kinase RIO2 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to RIOK2 (unknown origin) | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 8 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to full length recombinant human MAPK8 using ATF2 as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric sci... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| SNF-related serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 890 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human SNRK E97G/P116A mutant (1 to 505 residues) using KKLRRTLSFAEPG peptide as substrate incubated for 40 mins in pr... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Glycogen synthase kinase-3 alpha (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 870 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human GSK3alpha S449A mutant (2 to end residues) using YRRAAVPPSPSLSR peptide as substrate incubated for 40 mins in p... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Mitogen-activated protein kinase 10 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to full length recombinant human MAPK10 using peptide substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric sc... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Homeodomain-interacting protein kinase 1 (Homo sapiens (Human)) | BDBM50550127 (CHEMBL4781866) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human HIPK1 (158 to 555 residues) using myelin ba as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric ... | Citation and Details Article DOI: 10.1039/d0md00292e BindingDB Entry DOI: 10.7270/Q2251NSH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
