Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227177 ((R)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19294 (2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227171 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227180 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227167 ((S)-N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208662 ((R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208678 ((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227175 ((R)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208653 ((R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227181 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208688 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 108 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208665 ((R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-tr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227183 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227166 ((S)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19294 (2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227173 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208662 ((R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 275 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227182 ((R)-benzyl 3-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227178 ((S)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208645 ((R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-benzyl-4H-1,2,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208678 ((R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208688 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227169 ((S)-N-((S)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227179 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208653 ((R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227172 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 820 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50208665 ((R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-tr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 870 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227165 ((S)-N-(1-(4-(2,4-dimethoxybenzyl)-5-benzyl-4H-1,2,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227168 ((S)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-tr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227176 ((R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-tr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227164 ((S)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227170 ((S)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227174 ((S)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Displacement of [125I]His9-ghrelin from human GHSR1a receptor expressed in LLC PK1 cells | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227181 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Antagonist activity at human GHSR1a receptor expressed in CHO cells assessed as reduction of ghrelin-induced intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227177 ((R)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 75 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM19331 (CHEMBL266063 | N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227167 ((S)-N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227172 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 88 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227171 ((S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227169 ((S)-N-((S)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 440 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227175 ((R)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227166 ((S)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.58E+3 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227174 ((S)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Growth hormone secretagogue receptor type 1 (Homo sapiens (Human)) | BDBM50227180 ((R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxyb...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
CNRS-Université Montpellier I Curated by ChEMBL | Assay Description Agonist activity at human GHSR1a receptor expressed in CHO cells assessed as intracellular calcium mobilization | Bioorg Med Chem Lett 18: 164-8 (2008) Article DOI: 10.1016/j.bmcl.2007.10.113 BindingDB Entry DOI: 10.7270/Q2HM586C | |||||||||||
More data for this Ligand-Target Pair |