Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nucleotide-binding oligomerization domain-containing protein 2 (Homo sapiens (Human)) | BDBM50056694![]() (CHEMBL3326943) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 2 (Homo sapiens (Human)) | BDBM50056693![]() (CHEMBL3326942) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 2 (Homo sapiens (Human)) | BDBM50056692![]() (CHEMBL3326941) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 2 (Homo sapiens (Human)) | BDBM50056691![]() (CHEMBL3326924) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 2 (Homo sapiens (Human)) | BDBM50056690![]() (CHEMBL3326923) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 1 (Homo sapiens (Human)) | BDBM50056689![]() (CHEMBL3326922) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 1 (Homo sapiens (Human)) | BDBM50056694![]() (CHEMBL3326943) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 1 (Homo sapiens (Human)) | BDBM50056693![]() (CHEMBL3326942) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 1 (Homo sapiens (Human)) | BDBM50056692![]() (CHEMBL3326941) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 1 (Homo sapiens (Human)) | BDBM50056691![]() (CHEMBL3326924) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 1 (Homo sapiens (Human)) | BDBM50056690![]() (CHEMBL3326923) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD1 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nucleotide-binding oligomerization domain-containing protein 2 (Homo sapiens (Human)) | BDBM50056689![]() (CHEMBL3326922) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Antagonist activity at human NOD2 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liq... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056705![]() (CHEMBL3326944) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.01E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056704![]() (CHEMBL3326940) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.12E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056703![]() (CHEMBL3326939) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.65E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056702![]() (CHEMBL3326934) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.74E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056701![]() (CHEMBL3326933) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.61E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056700![]() (CHEMBL3326932) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.21E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056699![]() (CHEMBL3326931) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.57E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056698![]() (CHEMBL3326930) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.13E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056697![]() (CHEMBL3326925) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.16E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056696![]() (CHEMBL2270741) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.96E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056695![]() (CHEMBL3326918) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.23E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM50056706![]() (CHEMBL3326946) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Toll-like receptor 8 (Homo sapiens (Human)) | BDBM62988![]() ((1-butylbenzimidazol-2-yl)amine;hydrochloride | 1-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.30E+3 | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description Agonist activity at human TLR8 stably expressed in HEK293 cells co-expressing secreted alkaline phosphatase assessed as NF-kappaB induction by liquid... | J Med Chem 57: 7325-41 (2014) Article DOI: 10.1021/jm500701q BindingDB Entry DOI: 10.7270/Q2JS9S3S | |||||||||||
More data for this Ligand-Target Pair |