Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50537072 (CHEMBL440072) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a |
Tarveda Therapeutics Curated by ChEMBL | Assay Description Displacement of [125I]somatostatin from human SSTR4 expressed in CHO-K1 cell membranes after 120 mins | J Med Chem 62: 2708-2719 (2019) Article DOI: 10.1021/acs.jmedchem.8b02036 BindingDB Entry DOI: 10.7270/Q2NK3JJ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM81767 (15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | n/a |
ETH Zurich Curated by ChEMBL | Assay Description Binding assay at human somatostatin receptor 4 (hsst4) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand. | J Med Chem 44: 2460-8 (2001) Article DOI: 10.1021/jm010816q BindingDB Entry DOI: 10.7270/Q2C53PKS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50473329 (CHEMBL311789) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a |
ETH Zurich Curated by ChEMBL | Assay Description Binding assay at human somatostatin receptor 4 (hsst4) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand. | J Med Chem 44: 2460-8 (2001) Article DOI: 10.1021/jm010816q BindingDB Entry DOI: 10.7270/Q2C53PKS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098609 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 182 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098610 (10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 321 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098617 (10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 353 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098614 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 574 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098602 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098605 (10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098608 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098616 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098612 (10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098615 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098619 (10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50098603 (10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Tulane University Health Sciences Center Curated by ChEMBL | Assay Description Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4) | J Med Chem 44: 1416-21 (2001) BindingDB Entry DOI: 10.7270/Q2M044QS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50192018 (CHEMBL3350037) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.74E+3 | n/a | n/a | n/a | n/a | n/a |
ETH Zurich Curated by ChEMBL | Assay Description Binding assay at human somatostatin receptor 4 (hsst4) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand. | J Med Chem 44: 2460-8 (2001) Article DOI: 10.1021/jm010816q BindingDB Entry DOI: 10.7270/Q2C53PKS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50065452 (2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.63E+3 | n/a | n/a | n/a | n/a | n/a |
University of California at San Diego Curated by ChEMBL | Assay Description In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells. | J Med Chem 41: 2679-85 (1998) Article DOI: 10.1021/jm970393l BindingDB Entry DOI: 10.7270/Q2Z60N6X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50423462 (CHEMBL251835) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 3.63E+3 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Binding affinity to human recombinant sst4 receptor | Bioorg Med Chem Lett 18: 979-82 (2008) Article DOI: 10.1016/j.bmcl.2007.12.030 BindingDB Entry DOI: 10.7270/Q2WQ053B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50065451 (2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.17E+3 | n/a | n/a | n/a | n/a | n/a |
University of California at San Diego Curated by ChEMBL | Assay Description In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells. | J Med Chem 41: 2679-85 (1998) Article DOI: 10.1021/jm970393l BindingDB Entry DOI: 10.7270/Q2Z60N6X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50065450 (2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.68E+3 | n/a | n/a | n/a | n/a | n/a |
University of California at San Diego Curated by ChEMBL | Assay Description In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells. | J Med Chem 41: 2679-85 (1998) Article DOI: 10.1021/jm970393l BindingDB Entry DOI: 10.7270/Q2Z60N6X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50423465 (ERGOLINE) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Binding affinity to human recombinant sst4 receptor | Bioorg Med Chem Lett 18: 979-82 (2008) Article DOI: 10.1016/j.bmcl.2007.12.030 BindingDB Entry DOI: 10.7270/Q2WQ053B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50537061 (CHEMBL4527856) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 5.48E+3 | n/a | n/a | n/a | n/a | n/a |
Tarveda Therapeutics Curated by ChEMBL | Assay Description Displacement of [125I]somatostatin from human SSTR4 expressed in CHO-K1 cell membranes after 120 mins | J Med Chem 62: 2708-2719 (2019) Article DOI: 10.1021/acs.jmedchem.8b02036 BindingDB Entry DOI: 10.7270/Q2NK3JJ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50423458 (CHEMBL252232) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.62E+3 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Binding affinity to human recombinant sst4 receptor | Bioorg Med Chem Lett 18: 979-82 (2008) Article DOI: 10.1016/j.bmcl.2007.12.030 BindingDB Entry DOI: 10.7270/Q2WQ053B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50423464 (CHEMBL252231) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 8.13E+3 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Binding affinity to human recombinant sst4 receptor | Bioorg Med Chem Lett 18: 979-82 (2008) Article DOI: 10.1016/j.bmcl.2007.12.030 BindingDB Entry DOI: 10.7270/Q2WQ053B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50065453 ((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 8.91E+3 | n/a | n/a | n/a | n/a | n/a |
University of California at San Diego Curated by ChEMBL | Assay Description In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells. | J Med Chem 41: 2679-85 (1998) Article DOI: 10.1021/jm970393l BindingDB Entry DOI: 10.7270/Q2Z60N6X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50473330 (CHEMBL309948) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a |
ETH Zurich Curated by ChEMBL | Assay Description Binding assay at human somatostatin receptor 4 (hsst4) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand. | J Med Chem 44: 2460-8 (2001) Article DOI: 10.1021/jm010816q BindingDB Entry DOI: 10.7270/Q2C53PKS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50423297 (CHEMBL251541 | Obelin) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.51E+4 | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Binding affinity to human recombinant sst4 receptor | Bioorg Med Chem Lett 17: 3983-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.086 BindingDB Entry DOI: 10.7270/Q2XP7675 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Somatostatin receptor type 4 (Homo sapiens (Human)) | BDBM50473331 (CHEMBL420948) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | <1.00E+5 | n/a | n/a | n/a | n/a | n/a |
ETH Zurich Curated by ChEMBL | Assay Description Binding assay at human somatostatin receptor 4 (hsst4) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand. | J Med Chem 44: 2460-8 (2001) Article DOI: 10.1021/jm010816q BindingDB Entry DOI: 10.7270/Q2C53PKS | |||||||||||
More data for this Ligand-Target Pair |