Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363009 (CHEMBL1946412) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363013 (CHEMBL191539) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363006 (CHEMBL363989) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363004 (CHEMBL1946140) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50130735 ((7-Chloro-1,1-dioxo-1,4-dihydro-1lambda*6*-benzo[1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363007 (CHEMBL1946272) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362998 (CHEMBL1945810) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363002 (CHEMBL115565) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 760 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363003 (CHEMBL1946139) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.41E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363008 (CHEMBL1946410) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362992 (CHEMBL1946411) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363011 (CHEMBL189093) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.75E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362991 (CHEMBL1946273) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363001 (CHEMBL1946137) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363012 (CHEMBL1946759) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.98E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362995 (CHEMBL1945807) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362997 (CHEMBL1945809) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362990 (CHEMBL1946138) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363010 (CHEMBL1946414) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.93E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362993 (CHEMBL1944656) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363005 (CHEMBL1946270) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362990 (CHEMBL1946138) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362994 (CHEMBL1946760) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362993 (CHEMBL1944656) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362992 (CHEMBL1946411) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362991 (CHEMBL1946273) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50363000 (CHEMBL1946136) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.65E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362999 (CHEMBL1946134) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362996 (CHEMBL1945808) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.89E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-binding cassette sub-family C member 8 (Rattus norvegicus) | BDBM50362989 (CHEMBL1945806) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Li£ge Curated by ChEMBL | Assay Description Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretion | J Med Chem 54: 8353-61 (2011) Article DOI: 10.1021/jm200786z BindingDB Entry DOI: 10.7270/Q2WQ047Q | |||||||||||
More data for this Ligand-Target Pair |