Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463126 (CHEMBL4238599) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463135 (CHEMBL4243878) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463127 (CHEMBL4237402) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463138 (CHEMBL4240401) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463128 (CHEMBL4249055) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463140 (CHEMBL4240109) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463131 (CHEMBL4248559) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463134 (CHEMBL4246868) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463139 (CHEMBL4243533) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463130 (CHEMBL4247460) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463141 (CHEMBL4244986) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463129 (CHEMBL4245253) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463137 (CHEMBL4241092) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463136 (CHEMBL4248116) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463133 (CHEMBL4240576) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463132 (CHEMBL4250683) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463124 (CHEMBL4248050) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463125 (CHEMBL4242611) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formation | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463126 (CHEMBL4238599) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to His-tagged Myc (unknown origin) expressed in Escherichia coli BL21 by Bio-FET analysis | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Myc proto-oncogene protein (Homo sapiens (Human)) | BDBM50463128 (CHEMBL4249055) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Binding affinity to His-tagged Myc (unknown origin) expressed in Escherichia coli BL21 by Bio-FET analysis | Bioorg Med Chem 26: 4234-4239 (2018) Article DOI: 10.1016/j.bmc.2018.07.019 BindingDB Entry DOI: 10.7270/Q2FJ2KDB | |||||||||||
More data for this Ligand-Target Pair |