Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547480 (CHEMBL4790235) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 278 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547479 (CHEMBL4794290) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 393 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547491 (CHEMBL4784916) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 532 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547492 (CHEMBL4779693) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 538 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50078022 (CHEMBL3417402) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
Universit£ di Napoli"Federico II" Curated by ChEMBL | Assay Description Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by... | J Med Chem 58: 2135-48 (2015) Article DOI: 10.1021/jm501123r BindingDB Entry DOI: 10.7270/Q2X35055 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547481 (CHEMBL4777011) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 704 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547483 (CHEMBL4778142) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 719 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547487 (CHEMBL4761391) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 725 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547484 (CHEMBL4780328) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 809 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547490 (CHEMBL4756429) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 856 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547482 (CHEMBL4754714) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 874 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547489 (CHEMBL4758680) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 925 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547488 (CHEMBL4797324) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 967 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547493 (CHEMBL4776616) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 992 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547485 (CHEMBL4753330) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.14E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50547486 (CHEMBL4790418) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.22E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM50078015 (CHEMBL3417395) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.20E+3 | n/a | n/a | n/a | n/a |
Universit£ di Napoli"Federico II" Curated by ChEMBL | Assay Description Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by... | J Med Chem 58: 2135-48 (2015) Article DOI: 10.1021/jm501123r BindingDB Entry DOI: 10.7270/Q2X35055 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apoptosis regulator BAX (Homo sapiens (Human)) | BDBM19149 (CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01454 BindingDB Entry DOI: 10.7270/Q2N301J4 | |||||||||||
More data for this Ligand-Target Pair |