Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146893 (4-{(E)-2-[({[2,4-Dichloro-3-(4-ethoxy-2-methyl-qui...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146905 (4-{(E)-2-[({[2,4-Dichloro-3-(4-methoxy-2-methyl-qu...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146907 (5-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146895 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146899 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067281 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.510 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 in guinea pig ileum membrane | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146903 (CHEMBL98460 | N-[4-((E)-2-{[({2,4-Dichloro-3-[2-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.560 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067289 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.650 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146892 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.680 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146906 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.690 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146911 ((E)-N-[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2-ylm...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.830 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146897 (CHEMBL98292 | {4-[3-({2-[(E)-3-(6-Acetylamino-pyri...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.910 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067281 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146894 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-propoxy-qu...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146908 (4-{(E)-2-[({[2,4-Dichloro-3-(4-isopropoxy-2-methyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146902 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-[({2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146902 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-[({2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146901 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146891 (5-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146899 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146910 ((E)-N-[({2,4-Dichloro-3-[2-methyl-4-(pyridin-2-ylm...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146896 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[3-(1-benzy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146890 (CHEMBL540300 | {8-[2,6-Dichloro-3-(methyl-{2-[(E)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146900 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-[({2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146898 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylcarbamoylme...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067289 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146897 (CHEMBL98292 | {4-[3-({2-[(E)-3-(6-Acetylamino-pyri...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146900 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-[({2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146903 (CHEMBL98460 | N-[4-((E)-2-{[({2,4-Dichloro-3-[2-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the B2 receptor in guinea pig ileum membrane; | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146892 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146905 (4-{(E)-2-[({[2,4-Dichloro-3-(4-methoxy-2-methyl-qu...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146908 (4-{(E)-2-[({[2,4-Dichloro-3-(4-isopropoxy-2-methyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146890 (CHEMBL540300 | {8-[2,6-Dichloro-3-(methyl-{2-[(E)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146904 (4-{(E)-2-[({[2,4-Dichloro-3-(4-cyclopentyloxy-2-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146896 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[3-(1-benzy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146898 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylcarbamoylme...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146893 (4-{(E)-2-[({[2,4-Dichloro-3-(4-ethoxy-2-methyl-qui...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146909 (CHEMBL99978 | {8-[2,6-Dichloro-3-(methyl-{2-[3-(4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2 | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146904 (4-{(E)-2-[({[2,4-Dichloro-3-(4-cyclopentyloxy-2-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146894 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-propoxy-qu...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 77 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146909 (CHEMBL99978 | {8-[2,6-Dichloro-3-(methyl-{2-[3-(4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co. Ltd. Curated by ChEMBL | Assay Description Inhibition of [3H]BK (1.0 nM) binding to the human bradykinin receptor B2, expressed in CHO cells | J Med Chem 47: 2853-63 (2004) Article DOI: 10.1021/jm030468n BindingDB Entry DOI: 10.7270/Q2JM2BCM | |||||||||||
More data for this Ligand-Target Pair |