Affinity Data by PubMed id=16078826

PubMed code 16078826

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Progesterone receptor (Homo sapiens (Human))	BDBM50118694 (4-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]...) Show SMILES CC1(C)OC(=O)Nc2ccc(cc12)-c1coc(c1)C#N Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50118696 (5-(4,4-Dimethyl-2-oxo-1,4-dihydro-2H-benzo[d][1,3]...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50118700 (6-(3-Chloro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo...) Show SMILES CC1(C)OC(=O)Nc2ccc(cc12)-c1cccc(Cl)c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50066523 (2,2,4-Trimethyl-6-(3-nitro-phenyl)-1,2-dihydro-qui...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	41	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50121156 (5-(3-Chloro-phenyl)-3,3-dimethyl-1,3-dihydro-indol...) Show SMILES CC1(C)C(=O)Nc2ccc(cc12)-c1cccc(Cl)c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	66	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50105565 (6-(3-Chloro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...) Show SMILES CC(C)n1c2cc(ccc2[nH]c1=O)-c1cccc(Cl)c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	73	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50105566 (6-(3-Nitro-phenyl)-3H-benzothiazol-2-one \| CHEMBL3...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	84	n/a	n/a	n/a	n/a	n/a	n/a
Women's Health Research Institute Curated by ChEMBL					Assay Description Inhibition of human progesterone receptor				J Med Chem 48: 5092-5 (2005) Article DOI: 10.1021/jm050358b BindingDB Entry DOI: 10.7270/Q2FF3RXG
Women's Health Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%