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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28154 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | 120 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28138 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | 430 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28141 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | 360 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28152 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27 | n/a | 210 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28154 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29 | n/a | 370 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28142 (methyl (2S)-2-[(3-bromobenzene)sulfonyl]-2-[(2R)-7...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | 150 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28137 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 31 | n/a | 1.81E+3 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28141 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 49 | n/a | 1.35E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28139 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 56 | n/a | 160 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28139 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 62 | n/a | 1.07E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28149 (2-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 65 | n/a | 240 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28138 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 73 | n/a | 1.39E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28150 (2-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 83 | n/a | 92 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28155 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | 160 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28142 (methyl (2S)-2-[(3-bromobenzene)sulfonyl]-2-[(2R)-7...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | 850 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28137 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | 2.17E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28151 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | 76 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28134 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28147 ((2S)-2-(benzenesulfonyl)-2-[(2R)-7-chloro-1H,2H,3H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | 110 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28152 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | 1.09E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28150 (2-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 290 | n/a | 430 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28151 (5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | 890 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28131 (methyl (2S)-2-(benzenesulfonyl)-2-[(2R)-7-chloro-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | 250 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28145 (methyl (2S)-2-(benzenesulfonyl)-2-[(4R)-11-chloro-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | 370 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28148 (2-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 490 | n/a | 170 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28143 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 500 | n/a | 340 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28135 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 540 | n/a | 2.08E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28140 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 700 | n/a | 190 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28135 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | 1.53E+3 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28134 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 820 | n/a | 2.18E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28149 (2-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 920 | n/a | 1.50E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28131 (methyl (2S)-2-(benzenesulfonyl)-2-[(2R)-7-chloro-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | 1.60E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28140 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.21E+3 | n/a | 840 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28153 (methyl 5-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.63E+3 | n/a | 1.26E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28147 ((2S)-2-(benzenesulfonyl)-2-[(2R)-7-chloro-1H,2H,3H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.79E+3 | n/a | 1.09E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28136 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.25E+3 | n/a | 2.30E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28148 (2-[(S)-(benzenesulfonyl)[(2R)-7-chloro-1H,2H,3H,4H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | 770 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28145 (methyl (2S)-2-(benzenesulfonyl)-2-[(4R)-11-chloro-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.58E+3 | n/a | 4.23E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28146 ((2S)-2-(benzenesulfonyl)-2-[(2R)-7-chloro-1H,2H,3H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70E+3 | n/a | 1.55E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28132 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.30E+3 | n/a | 370 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28132 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.30E+3 | n/a | 5.81E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28136 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.42E+3 | n/a | 3.16E+3 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28146 ((2S)-2-(benzenesulfonyl)-2-[(2R)-7-chloro-1H,2H,3H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.87E+3 | n/a | 400 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28144 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.95E+3 | n/a | 270 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28144 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.22E+4 | n/a | 2.75E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28143 (methyl (2S)-2-[(2R)-7-chloro-1H,2H,3H,4H-cyclopent...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | 1.07E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-beta (Homo sapiens (Human)) | BDBM28133 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.12E+4 | n/a | >4.00E+4 | n/a | n/a | n/a | n/a |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Oxysterols receptor LXR-alpha (Homo sapiens (Human)) | BDBM28133 (methyl (2S)-2-[(2R)-6-chloro-2,3,4,9-tetrahydro-1H...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.79E+4 | n/a | 5.80E+3 | n/a | n/a | 7.4 | 22 |
F. Hoffmann-La Roche Ltd | Assay Description LXR receptor binding assays were performed in 96-well plates. For each well reaction, GST-LXR-LBD fusion proteins were bound to SPA beads, and radiol... | Bioorg Med Chem Lett 19: 1654-7 (2009) Article DOI: 10.1016/j.bmcl.2009.01.109 BindingDB Entry DOI: 10.7270/Q2BK19PN | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
