Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29546 (benzimidazolone scaffold, 15d) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 3.40 | -50.3 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29548 (benzimidazolone scaffold, 15f) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | -48.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29549 (benzimidazolone scaffold, 15g) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29554 (benzimidazolone scaffold, 15m) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29553 (benzimidazolone scaffold, 15k) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29552 (benzimidazolone scaffold, 15j) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 12 | -47.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29551 (benzimidazolone scaffold, 15i) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29540 (benzimidazolone scaffold, 8h) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 22 | -45.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29544 (benzimidazolone scaffold, 15b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 25 | -45.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29541 (benzimidazolone scaffold, 17d) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 26 | -45.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29545 (benzimidazolone scaffold, 15c) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 26 | -45.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29548 (benzimidazolone scaffold, 15f) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29550 (benzimidazolone scaffold, 15h) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 33 | -44.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29542 (benzimidazolone scaffold, 17f) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 36 | -44.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29550 (benzimidazolone scaffold, 15h) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29546 (benzimidazolone scaffold, 15d) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29547 (benzimidazolone scaffold, 15e) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 48 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29551 (benzimidazolone scaffold, 15i) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 48 | -43.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29553 (benzimidazolone scaffold, 15k) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 66 | -42.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29552 (benzimidazolone scaffold, 15j) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29547 (benzimidazolone scaffold, 15e) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 84 | -42.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29537 (benzimidazolone scaffold, 8e) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 168 | -40.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29541 (benzimidazolone scaffold, 17d) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 168 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29539 (benzimidazolone scaffold, 8g) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 182 | -40.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29545 (benzimidazolone scaffold, 15c) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 243 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29542 (benzimidazolone scaffold, 17f) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 267 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29549 (benzimidazolone scaffold, 15g) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 269 | -39.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29540 (benzimidazolone scaffold, 8h) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 296 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29536 (benzimidazolone scaffold, 8d) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 340 | -38.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29538 (benzimidazolone scaffold, 8f) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 375 | -38.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29543 (benzimidazolone scaffold, 15a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 392 | -38.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29554 (benzimidazolone scaffold, 15m) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 454 | -37.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29533 (benzimidazolone scaffold, 8a) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 467 | -37.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29536 (benzimidazolone scaffold, 8d) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 566 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29534 (benzimidazolone scaffold, 8b) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 636 | -36.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM29535 (benzimidazolone scaffold, 8c) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 646 | -36.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 37 |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29535 (benzimidazolone scaffold, 8c) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 864 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29534 (benzimidazolone scaffold, 8b) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 902 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29543 (benzimidazolone scaffold, 15a) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 1.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29533 (benzimidazolone scaffold, 8a) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29544 (benzimidazolone scaffold, 15b) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 1.84E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29537 (benzimidazolone scaffold, 8e) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29539 (benzimidazolone scaffold, 8g) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (Homo sapiens (Human)) | BDBM29538 (benzimidazolone scaffold, 8f) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
CNRS | Assay Description Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b... | Bioorg Med Chem Lett 19: 1600-3 (2009) Article DOI: 10.1016/j.bmcl.2009.02.008 BindingDB Entry DOI: 10.7270/Q2KS6PW1 | |||||||||||
More data for this Ligand-Target Pair |