Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50060728 ((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 20.9 | n/a | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50394978 (CHEMBL573297) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50336912 (Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 379 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50394976 (CHEMBL2165922) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 41.7 | n/a | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50394978 (CHEMBL573297) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 527 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50394975 (CHEMBL2165921) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.62E+3 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50394977 (CHEMBL583068) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.37E+3 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50394977 (CHEMBL583068) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.19E+3 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM86143 (L-Val-L-Pro-L-Asn-L-Leu-L-Pro-L-Gln-L-Arg-L-Phe-NH...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50060728 ((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 233 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50394975 (CHEMBL2165921) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.66E+3 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM86143 (L-Val-L-Pro-L-Asn-L-Leu-L-Pro-L-Gln-L-Arg-L-Phe-NH...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 2 (Homo sapiens (Human)) | BDBM50394976 (CHEMBL2165922) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 298 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide FF receptor 1 (Homo sapiens (Human)) | BDBM50336912 (Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 71 | n/a | n/a | n/a | n/a |
Leipzig University Curated by ChEMBL | Assay Description Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ... | J Med Chem 55: 6124-36 (2012) Article DOI: 10.1021/jm300535s BindingDB Entry DOI: 10.7270/Q26974PV | |||||||||||
More data for this Ligand-Target Pair |