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PubMed code 23357035

Compile data set for download or QSAR
Found 19 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429385
PNG
(CHEMBL2336756)
Show SMILES COc1cc2nc(nc(Nc3ccc(cc3F)S(C)(=O)=O)c2cc1OC)N1CCC2CCC(C1)N2Cc1ccccc1 |TLB:6:26:34:30.31,35:34:33.26.27.28:30.31|
Show InChI InChI=1S/C31H34FN5O4S/c1-40-28-16-24-27(17-29(28)41-2)34-31(35-30(24)33-26-12-11-23(15-25(26)32)42(3,38)39)36-14-13-21-9-10-22(19-36)37(21)18-20-7-5-4-6-8-20/h4-8,11-12,15-17,21-22H,9-10,13-14,18-19H2,1-3H3,(H,33,34,35)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429393
PNG
(CHEMBL2336765)
Show SMILES COc1cc2nc(OC3CCN(CC3)C(=O)OC(C)(C)C)nc(Nc3ccc(cc3F)S(C)(=O)=O)c2cc1OC
Show InChI InChI=1S/C27H33FN4O7S/c1-27(2,3)39-26(33)32-11-9-16(10-12-32)38-25-30-21-15-23(37-5)22(36-4)14-18(21)24(31-25)29-20-8-7-17(13-19(20)28)40(6,34)35/h7-8,13-16H,9-12H2,1-6H3,(H,29,30,31)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429398
PNG
(CHEMBL2336759)
Show SMILES COc1cc2nc(nc(Nc3ccc(cc3F)S(C)(=O)=O)c2cc1OC)N1CCC2CCC(C1)N2C(=O)OC(C)(C)C |TLB:35:34:33.26.27.28:30.31,6:26:34:30.31|
Show InChI InChI=1S/C29H36FN5O6S/c1-29(2,3)41-28(36)35-17-7-8-18(35)16-34(12-11-17)27-32-23-15-25(40-5)24(39-4)14-20(23)26(33-27)31-22-10-9-19(13-21(22)30)42(6,37)38/h9-10,13-15,17-18H,7-8,11-12,16H2,1-6H3,(H,31,32,33)
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n/an/an/an/a 1.00E+3n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429388
PNG
(CHEMBL2336771)
Show SMILES COc1cc2nc(NCC3CC4CCC(C3)N4C(=O)OC(C)(C)C)nc(Nc3ccc(cc3)S(C)(=O)=O)c2cc1OC |THB:8:9:16:12.13|
Show InChI InChI=1S/C30H39N5O6S/c1-30(2,3)41-29(36)35-20-9-10-21(35)14-18(13-20)17-31-28-33-24-16-26(40-5)25(39-4)15-23(24)27(34-28)32-19-7-11-22(12-8-19)42(6,37)38/h7-8,11-12,15-16,18,20-21H,9-10,13-14,17H2,1-6H3,(H2,31,32,33,34)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429394
PNG
(CHEMBL2336764)
Show SMILES COc1cc2nc(Nc3ccc(cc3F)S(C)(=O)=O)nc(OC3CCN(CC3)C(=O)OC(C)(C)C)c2cc1OC
Show InChI InChI=1S/C27H33FN4O7S/c1-27(2,3)39-26(33)32-11-9-16(10-12-32)38-24-18-14-22(36-4)23(37-5)15-21(18)30-25(31-24)29-20-8-7-17(13-19(20)28)40(6,34)35/h7-8,13-16H,9-12H2,1-6H3,(H,29,30,31)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429395
PNG
(CHEMBL2336762)
Show SMILES COc1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)nc(OCC3CCN(CC3)C(=O)OC(C)(C)C)c2cc1OC
Show InChI InChI=1S/C28H36N4O7S/c1-28(2,3)39-27(33)32-13-11-18(12-14-32)17-38-25-21-15-23(36-4)24(37-5)16-22(21)30-26(31-25)29-19-7-9-20(10-8-19)40(6,34)35/h7-10,15-16,18H,11-14,17H2,1-6H3,(H,29,30,31)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429396
PNG
(CHEMBL2336761)
Show SMILES COc1cc2nc(OC3CCN(CC3)C(=O)OC(C)(C)C)nc(Nc3ccc(cc3)S(C)(=O)=O)c2cc1OC
Show InChI InChI=1S/C27H34N4O7S/c1-27(2,3)38-26(32)31-13-11-18(12-14-31)37-25-29-21-16-23(36-5)22(35-4)15-20(21)24(30-25)28-17-7-9-19(10-8-17)39(6,33)34/h7-10,15-16,18H,11-14H2,1-6H3,(H,28,29,30)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429397
PNG
(CHEMBL2336760)
Show SMILES COc1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)nc(OC3CCN(CC3)C(=O)OC(C)(C)C)c2cc1OC
Show InChI InChI=1S/C27H34N4O7S/c1-27(2,3)38-26(32)31-13-11-18(12-14-31)37-24-20-15-22(35-4)23(36-5)16-21(20)29-25(30-24)28-17-7-9-19(10-8-17)39(6,33)34/h7-10,15-16,18H,11-14H2,1-6H3,(H,28,29,30)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM29080
PNG
(CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA...)
Show SMILES CCCCCCCC\C=C/CCCCCCCC(=O)NCCO
Show InChI InChI=1S/C20H39NO2/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-16-17-20(23)21-18-19-22/h9-10,22H,2-8,11-19H2,1H3,(H,21,23)/b10-9-
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n/an/an/an/a 2.20E+3n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429392
PNG
(CHEMBL2336766)
Show SMILES COc1cc2nc(Nc3ccc(cc3F)S(C)(=O)=O)nc(OCC3CCN(CC3)C(=O)OC(C)(C)C)c2cc1OC
Show InChI InChI=1S/C28H35FN4O7S/c1-28(2,3)40-27(34)33-11-9-17(10-12-33)16-39-25-19-14-23(37-4)24(38-5)15-22(19)31-26(32-25)30-21-8-7-18(13-20(21)29)41(6,35)36/h7-8,13-15,17H,9-12,16H2,1-6H3,(H,30,31,32)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429383
PNG
(CHEMBL2336758)
Show SMILES COc1cc2nc(nc(Nc3ccc(cc3)S(C)(=O)=O)c2cc1OC)N1CCC2CCC(C1)N2C(=O)OC(C)(C)C |TLB:34:33:32.25.26.27:29.30,6:25:33:29.30|
Show InChI InChI=1S/C29H37N5O6S/c1-29(2,3)40-28(35)34-19-9-10-20(34)17-33(14-13-19)27-31-23-16-25(39-5)24(38-4)15-22(23)26(32-27)30-18-7-11-21(12-8-18)41(6,36)37/h7-8,11-12,15-16,19-20H,9-10,13-14,17H2,1-6H3,(H,30,31,32)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429386
PNG
(CHEMBL2336755)
Show SMILES COc1cc2nc(nc(Nc3ccc(cc3)S(C)(=O)=O)c2cc1OC)N1CCC2CCC(C1)N2Cc1ccccc1 |TLB:6:25:33:29.30,34:33:32.25.26.27:29.30|
Show InChI InChI=1S/C31H35N5O4S/c1-39-28-17-26-27(18-29(28)40-2)33-31(34-30(26)32-22-9-13-25(14-10-22)41(3,37)38)35-16-15-23-11-12-24(20-35)36(23)19-21-7-5-4-6-8-21/h4-10,13-14,17-18,23-24H,11-12,15-16,19-20H2,1-3H3,(H,32,33,34)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429389
PNG
(CHEMBL2336770)
Show SMILES COc1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)nc(NCC3CC4CCC(C3)N4C(=O)OC(C)(C)C)c2cc1OC |THB:21:22:29:25.26|
Show InChI InChI=1S/C30H39N5O6S/c1-30(2,3)41-29(36)35-20-9-10-21(35)14-18(13-20)17-31-27-23-15-25(39-4)26(40-5)16-24(23)33-28(34-27)32-19-7-11-22(12-8-19)42(6,37)38/h7-8,11-12,15-16,18,20-21H,9-10,13-14,17H2,1-6H3,(H2,31,32,33,34)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429390
PNG
(CHEMBL2336768)
Show SMILES COc1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)nc(NC3CC4CCC(C3)N4C(=O)OC(C)(C)C)c2cc1OC |TLB:20:21:28:24.25|
Show InChI InChI=1S/C29H37N5O6S/c1-29(2,3)40-28(35)34-19-9-10-20(34)14-18(13-19)30-26-22-15-24(38-4)25(39-5)16-23(22)32-27(33-26)31-17-7-11-21(12-8-17)41(6,36)37/h7-8,11-12,15-16,18-20H,9-10,13-14H2,1-6H3,(H2,30,31,32,33)
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Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429384
PNG
(CHEMBL2336757)
Show SMILES COc1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)nc(N3CCC4CCC(C3)N4C(=O)OC(C)(C)C)c2cc1OC |TLB:29:28:27.20.21.22:24.25,THB:19:20:28:24.25|
Show InChI InChI=1S/C29H37N5O6S/c1-29(2,3)40-28(35)34-19-9-10-20(34)17-33(14-13-19)26-22-15-24(38-4)25(39-5)16-23(22)31-27(32-26)30-18-7-11-21(12-8-18)41(6,36)37/h7-8,11-12,15-16,19-20H,9-10,13-14,17H2,1-6H3,(H,30,31,32)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429399
PNG
(CHEMBL2336753)
Show SMILES COc1cc2nc(NCC3CC4CCC(C3)N4C(=O)OC(C)(C)C)nc(Nc3ccc(cc3F)S(C)(=O)=O)c2cc1OC |THB:8:9:16:12.13|
Show InChI InChI=1S/C30H38FN5O6S/c1-30(2,3)42-29(37)36-18-7-8-19(36)12-17(11-18)16-32-28-34-24-15-26(41-5)25(40-4)14-21(24)27(35-28)33-23-10-9-20(13-22(23)31)43(6,38)39/h9-10,13-15,17-19H,7-8,11-12,16H2,1-6H3,(H2,32,33,34,35)
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n/an/an/an/a 1.00E+3n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429400
PNG
(CHEMBL2336769)
Show SMILES COc1cc2nc(NC3CC4CCC(C3)N4C(=O)OC(C)(C)C)nc(Nc3ccc(cc3F)S(C)(=O)=O)c2cc1OC |TLB:7:8:15:11.12|
Show InChI InChI=1S/C29H36FN5O6S/c1-29(2,3)41-28(36)35-17-7-8-18(35)12-16(11-17)31-27-33-23-15-25(40-5)24(39-4)14-20(23)26(34-27)32-22-10-9-19(13-21(22)30)42(6,37)38/h9-10,13-18H,7-8,11-12H2,1-6H3,(H2,31,32,33,34)
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n/an/an/an/a 1.00E+3n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429387
PNG
(CHEMBL2336754)
Show SMILES COc1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)nc(N3CCC4CCC(C3)N4Cc3ccccc3)c2cc1OC |TLB:29:28:27.20.21.22:24.25,THB:19:20:28:24.25|
Show InChI InChI=1S/C31H35N5O4S/c1-39-28-17-26-27(18-29(28)40-2)33-31(32-22-9-13-25(14-10-22)41(3,37)38)34-30(26)35-16-15-23-11-12-24(20-35)36(23)19-21-7-5-4-6-8-21/h4-10,13-14,17-18,23-24H,11-12,15-16,19-20H2,1-3H3,(H,32,33,34)
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n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50429391
PNG
(CHEMBL2336767)
Show SMILES COc1cc2nc(OCC3CCN(CC3)C(=O)OC(C)(C)C)nc(Nc3ccc(cc3F)S(C)(=O)=O)c2cc1OC
Show InChI InChI=1S/C28H35FN4O7S/c1-28(2,3)40-27(34)33-11-9-17(10-12-33)16-39-26-31-22-15-24(38-5)23(37-4)14-19(22)25(32-26)30-21-8-7-18(13-20(21)29)41(6,35)36/h7-8,13-15,17H,9-12,16H2,1-6H3,(H,30,31,32)
PDB

UniProtKB/SwissProt

antibodypedia
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CHEMBL
PC cid
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UniChem

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PubMed
n/an/an/an/a>1.00E+4n/an/an/an/a



Kangwon National University

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 60 mins

Bioorg Med Chem 21: 1349-56 (2013)


Article DOI: 10.1016/j.bmc.2012.12.013
BindingDB Entry DOI: 10.7270/Q2ZG6TKZ
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%