Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50033969 (3-(2,4-Difluoro-phenyl)-1-[5-(4,5-diphenyl-1H-imid...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450322 (CHEMBL431934) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of ACYL CoA:Cholesterol Acyltransferase (ACAT) in rat hepatic microsomes was measured by using AIV assay | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450338 (CHEMBL416816) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450330 (CHEMBL295251) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50037632 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(4-phenyl-1H...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 490 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450335 (CHEMBL416998) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450327 (CHEMBL300518) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450313 (CHEMBL46174) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 810 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450333 (CHEMBL48094) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50033969 (3-(2,4-Difluoro-phenyl)-1-[5-(4,5-diphenyl-1H-imid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450323 (CHEMBL46017) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450324 (CHEMBL45913) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 1.53E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50037632 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(4-phenyl-1H...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450329 (CHEMBL295079) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450314 (CHEMBL417187) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450323 (CHEMBL46017) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 2.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450320 (CHEMBL49001) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450337 (CHEMBL291197) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 2.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450313 (CHEMBL46174) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 2.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450336 (CHEMBL45964) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 2.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450322 (CHEMBL431934) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450320 (CHEMBL49001) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50037630 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(1H-imidazol...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 2.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450337 (CHEMBL291197) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 3.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450335 (CHEMBL416998) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450332 (CHEMBL45740) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450327 (CHEMBL300518) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 3.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450343 (CHEMBL432696) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50037635 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(1-methyl-4,...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 3.56E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450324 (CHEMBL45913) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450318 (CHEMBL49398) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50037635 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(1-methyl-4,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450341 (CHEMBL297676) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450342 (CHEMBL295286) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450315 (CHEMBL46387) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450336 (CHEMBL45964) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450342 (CHEMBL295286) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450344 (CHEMBL289648) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450328 (CHEMBL44610) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450332 (CHEMBL45740) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 4.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450315 (CHEMBL46387) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450339 (CHEMBL45184) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 4.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450334 (CHEMBL49957) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450325 (CHEMBL50554) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450340 (CHEMBL48106) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450338 (CHEMBL416816) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 5.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450318 (CHEMBL49398) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 5.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50037630 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(1H-imidazol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50037643 (3-(2,4-Difluoro-phenyl)-1-[5-(1,4-diphenyl-1H-imid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 6.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450321 (CHEMBL45915) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 6.53E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450319 (CHEMBL47863) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 6.96E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450326 (CHEMBL45484) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 7.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450328 (CHEMBL44610) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 7.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450326 (CHEMBL45484) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 7.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50037643 (3-(2,4-Difluoro-phenyl)-1-[5-(1,4-diphenyl-1H-imid...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 7.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450314 (CHEMBL417187) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 8.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450316 (CHEMBL297991) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 9.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450331 (CHEMBL49215) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 9.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450330 (CHEMBL295251) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 1.06E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450341 (CHEMBL297676) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450325 (CHEMBL50554) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450317 (CHEMBL46318) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 1.91E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450317 (CHEMBL46318) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.37E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450316 (CHEMBL297991) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450340 (CHEMBL48106) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.73E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450334 (CHEMBL49957) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 2.97E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450343 (CHEMBL432696) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50037645 (3-(2,4-Difluoro-phenyl)-1-heptyl-1-[5-(1,4,5-triph...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 5.45E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450329 (CHEMBL295079) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 6.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Mus musculus) | BDBM50450344 (CHEMBL289648) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 7.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description Inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in J774 Macrophage cell culture by using J774 assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50450331 (CHEMBL49215) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | n/a | n/a | 7.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
The DuPont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase (ACAT) in rat hepatic microsomes by using AIV assay. | Bioorg Med Chem Lett 5: 167-72 (1995) BindingDB Entry DOI: 10.7270/Q2Z03833 | |||||||||||
More data for this Ligand-Target Pair |