| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin E2 receptor EP2 subtype |
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| Ligand | BDBM50213909 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_456180 (CHEMBL888190) |
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| Ki | 3000±n/a nM |
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| Citation |  Sandham, DA; Aldcroft, C; Baettig, U; Barker, L; Beer, D; Bhalay, G; Brown, Z; Dubois, G; Budd, D; Bidlake, L; Campbell, E; Cox, B; Everatt, B; Harrison, D; Leblanc, CJ; Manini, J; Profit, R; Stringer, R; Thompson, KS; Turner, KL; Tweed, MF; Walker, C; Watson, SJ; Whitebread, S; Willis, J; Williams, G; Wilson, C 2-Cycloalkyl phenoxyacetic acid CRTh2 receptor antagonists. Bioorg Med Chem Lett17:4347-50 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin E2 receptor EP2 subtype |
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| Name: | Prostaglandin E2 receptor EP2 subtype |
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| Synonyms: | PE2R2_HUMAN | PGE receptor EP2 subtype | PTGER2 | Prostaglandin E2 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype | Prostanoid EP2 Receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 39775.71 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P43116 |
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| Residue: | 358 |
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| Sequence: | MGNASNDSQSEDCETRQWLPPGESPAISSVMFSAGVLGNLIALALLARRWRGDVGCSAGR
RSSLSLFHVLVTELVFTDLLGTCLISPVVLASYARNQTLVALAPESRACTYFAFAMTFFS
LATMLMLFAMALERYLSIGHPYFYQRRVSRSGGLAVLPVIYAVSLLFCSLPLLDYGQYVQ
YCPGTWCFIRHGRTAYLQLYATLLLLLIVSVLACNFSVILNLIRMHRRSRRSRCGPSLGS
GRGGPGARRRGERVSMAEETDHLILLAIMTITFAVCSLPFTIFAYMNETSSRKEKWDLQA
LRFLSINSIIDPWVFAILRPPVLRLMRSVLCCRISLRTQDATQTSCSTQSDASKQADL
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| BDBM50213909 |
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| n/a |
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| Name | BDBM50213909 |
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| Synonyms: | 2-(4-chloro-2-cyclohexylphenoxy)acetic acid | CHEMBL245908 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H17ClO3 |
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| Mol. Mass. | 268.736 |
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| SMILES | OC(=O)COc1ccc(Cl)cc1C1CCCCC1 |
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| Structure | 
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