| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin D2 receptor |
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| Ligand | BDBM50213907 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_456179 (CHEMBL888189) |
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| Ki | 6400±n/a nM |
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| Citation |  Sandham, DA; Aldcroft, C; Baettig, U; Barker, L; Beer, D; Bhalay, G; Brown, Z; Dubois, G; Budd, D; Bidlake, L; Campbell, E; Cox, B; Everatt, B; Harrison, D; Leblanc, CJ; Manini, J; Profit, R; Stringer, R; Thompson, KS; Turner, KL; Tweed, MF; Walker, C; Watson, SJ; Whitebread, S; Willis, J; Williams, G; Wilson, C 2-Cycloalkyl phenoxyacetic acid CRTh2 receptor antagonists. Bioorg Med Chem Lett17:4347-50 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin D2 receptor |
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| Name: | Prostaglandin D2 receptor |
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| Synonyms: | PD2R_HUMAN | PTGDR | Prostaglandin D2 | Prostaglandin D2 receptor | Prostanoid DP receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 40288.87 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q13258 |
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| Residue: | 359 |
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| Sequence: | MKSPFYRCQNTTSVEKGNSAVMGGVLFSTGLLGNLLALGLLARSGLGWCSRRPLRPLPSV
FYMLVCGLTVTDLLGKCLLSPVVLAAYAQNRSLRVLAPALDNSLCQAFAFFMSFFGLSST
LQLLAMALECWLSLGHPFFYRRHITLRLGALVAPVVSAFSLAFCALPFMGFGKFVQYCPG
TWCFIQMVHEEGSLSVLGYSVLYSSLMALLVLATVLCNLGAMRNLYAMHRRLQRHPRSCT
RDCAEPRADGREASPQPLEELDHLLLLALMTVLFTMCSLPVIYRAYYGAFKDVKEKNRTS
EEAEDLRALRFLSVISIVDPWIFIIFRSPVFRIFFHKIFIRPLRYRSRCSNSTNMESSL
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| BDBM50213907 |
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| n/a |
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| Name | BDBM50213907 |
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| Synonyms: | (3-cyclohexyl-4'-fluoro-biphenyl-4-yloxy)-acetic acid | CHEMBL429470 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H21FO3 |
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| Mol. Mass. | 328.3773 |
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| SMILES | OC(=O)COc1ccc(cc1C1CCCCC1)-c1ccc(F)cc1 |
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| Structure | 
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