Reaction Details |
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Target | Mitogen-activated protein kinase 11 |
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Ligand | BDBM16526 |
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Substrate/Competitor | biotinylated GST-ATF2 |
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Meas. Tech. | Enzyme Inhibition Scintillation Proximity Assay |
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IC50 | 41±n/a nM |
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Citation | Natarajan, SR; Heller, ST; Nam, K; Singh, SB; Scapin, G; Patel, S; Thompson, JE; Fitzgerald, CE; O'Keefe, SJ p38 MAP kinase inhibitors. Part 6: 2-arylpyridazin-3-ones as templates for inhibitor design. Bioorg Med Chem Lett16:5809-13 (2006) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Mitogen-activated protein kinase 11 |
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Name: | Mitogen-activated protein kinase 11 |
Synonyms: | MAP Kinase p38 beta | MK11_MOUSE | Mapk11 | Mitogen-activated protein kinase 11 | Mitogen-activated protein kinase p38 beta | Prkm11 | p38B |
Type: | Enzyme |
Mol. Mass.: | 41390.66 |
Organism: | Mus musculus (mouse) |
Description: | Q9WUI1 |
Residue: | 364 |
Sequence: | MSGPRAGFYRQELNKTVWEVPQRLQGLRPVGSGAYGSVCSAYDARLRQKVAVKKLSRPFQ
SLIHARRTYRELRLLKHLKHENVIGLLDVFTPATSIEDFSEVYLVTTLMGADLNNIVKCQ
ALSDEHVQFLVYQLLRGLKYIHSAGIIHRDLKPSNVAVNEDCELRILDFGLARQADEEMT
GYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLQGKALFPGNDYIDQLKRIMEVVG
TPSPEVLAKISSEHARTYIQSLPPMPQKDLSSVFHGANPLAIDLLGRMLVLDSDQRVSAA
EALAHAYFSQYHDPDDEPEAEPYDESVEAKERTLEEWKELTYQEVLSFKPLEPSQLPGTH
EIEQ
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BDBM16526 |
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biotinylated GST-ATF2 |
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Name: | biotinylated GST-ATF2 |
Synonyms: | ATF-2-GST | ATF2 | Activating transcription factor 2 | Activating transcription factor 2-GST fusion | GST-ATF2 | biotinylated ATF2 substrate | biotinylated activating transcription factor 2 |
Type: | Other Protein Type |
Mol. Mass.: | 12237.77 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 109 |
Sequence: | MSDDKPFLCTAPGCGQRFTNEDHLAVHKHKHEMTLKFGPARNDSVIVADQTPTPTRFLKN
CEEVGLFNELASPFENEFKKASEDDIKKMPLDLSPLATPIIRSKIEEPS
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