| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50120060 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_149317 |
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| Ki | 1151±n/a nM |
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| Citation |  Roy, C; Li, T; Krasik, P; Gilbert, MJ; Pelletier, C; Gagnon, D; Robert, E; Ducharme, J; Storer, R; Lavallée, JF Synthesis and structure--activity relationship of novel aminotetralin derivatives with high micro selective opioid affinity. Bioorg Med Chem Lett12:3141-3 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44789.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35372 |
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| Residue: | 400 |
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| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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|
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| BDBM50120060 |
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| n/a |
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| Name | BDBM50120060 |
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| Synonyms: | 7-Amino-6-methanesulfonyl-8,8-dimethyl-5,6,7,8-tetrahydro-naphthalen-2-ol | CHEMBL107442 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H19NO3S |
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| Mol. Mass. | 269.36 |
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| SMILES | CC1(C)[C@H](N)[C@@H](Cc2ccc(O)cc12)S(C)(=O)=O |
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| Structure | 
|
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