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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Neuropeptide Y receptor type 5 | ||
| Ligand | BDBM50353147 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_768586 (CHEMBL1832605) | ||
| Ki | 8.4±n/a nM | ||
| Citation |  Wu, L; Lu, K; Desai, M; Packiarajan, M; Joshi, A; Marzabadi, MR; Jubian, V; Andersen, K; Chandrasena, G; Boyle, NJ; Walker, MW N-Heteroaryl glycinamides and glycinamines as potent NPY5 antagonists. Bioorg Med Chem Lett21:5573-6 (2011) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Neuropeptide Y receptor type 5 | |||
| Name: | Neuropeptide Y receptor type 5 | ||
| Synonyms: | NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPY5R_HUMAN | NPYR5 | NPYY5 | Neuropeptide Y receptor type 5 | Neuropeptide Y receptor type 5 ( NPY Y5) | Y5 receptor | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 50746.64 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | Q15761 | ||
| Residue: | 445 | ||
| Sequence: |
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| BDBM50353147 | |||
| n/a | |||
| Name | BDBM50353147 | ||
| Synonyms: | CHEMBL1829319 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C20H28FN3O5S | ||
| Mol. Mass. | 441.517 | ||
| SMILES | CC(C)S(=O)(=O)NC[C@H]1CC[C@@H](CC1)NC(=O)CN1C(=O)COc2cc(F)ccc12 |r,wU:11.14,wD:8.7,(10.22,-.38,;8.88,.4,;8.89,1.94,;7.55,-.37,;6.77,-1.7,;8.31,-1.7,;6.22,.4,;4.88,-.36,;3.55,.41,;3.55,1.95,;2.22,2.73,;.89,1.95,;.89,.41,;2.21,-.36,;-.45,2.72,;-1.78,1.95,;-1.78,.41,;-3.11,2.71,;-4.45,1.94,;-4.45,.4,;-3.12,-.37,;-5.78,-.37,;-7.11,.4,;-7.11,1.93,;-8.45,2.7,;-8.45,4.25,;-9.78,5.02,;-7.12,5.02,;-5.79,4.25,;-5.78,2.7,)| | ||
| Structure | 
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