| Reaction Details |
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 | Report a problem with these data |
| Target | Histamine H2 receptor |
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| Ligand | BDBM22881 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_85683 |
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| Kd | 11482±n/a nM |
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| Citation |  van der Goot, H; Eriks, JC; Leurs, R; Timmerman, H Amselamine, a new selective histamine H2-receptor agonist Bioorg Med Chem Lett4:1913-1916 (1994) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Histamine H2 receptor |
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| Name: | Histamine H2 receptor |
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| Synonyms: | Gastric receptor I | H2R | HISTAMINE H2 | HRH2_RAT | Hrh2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40269.37 |
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| Organism: | RAT |
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| Description: | HISTAMINE H2 HRH2 RAT::P25102 |
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| Residue: | 358 |
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| Sequence: | MEPNGTVHSCCLDSMALKVTISVVLTTLILITIAGNVVVCLAVSLNRRLRSLTNCFIVSL
AATDLLLGLLVLPFSAIYQLSFTWSFGHVFCNIYTSLDVMLCTASILNLFMISLDRYCAV
TDPLRYPVLVTPVRVAISLVFIWVISITLSFLSIHLGWNSRNGTRGGNDTFKCKVQVNEV
YGLVDGLVTFYLPLLIMCVTYYRIFKIAREQAKRINHISSWKAATIREHKATVTLAAVMG
AFIICWFPYFTAFVYRGLRGDDAINEAVEGIVLWLGYANSALNPILYAALNRDFRTAYQQ
LFHCKFASHNSHKTSLRLNNSLLPRSQSREGRWQEEKPLKLQVWSGTELTHPQGNPIR
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| BDBM22881 |
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| n/a |
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| Name | BDBM22881 |
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| Synonyms: | 5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-amine | Amthamine | CHEMBL554964 |
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| Type | Small organic molecule |
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| Emp. Form. | C6H11N3S |
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| Mol. Mass. | 157.237 |
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| SMILES | Cc1nc(N)sc1CCN |
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| Structure | 
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