| Reaction Details |
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 | Report a problem with these data |
| Target | Urotensin-2 |
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| Ligand | BDBM50416336 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_643307 (CHEMBL1177478) |
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| EC50 | 134.9±n/a nM |
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| Citation |  Lehmann, F; Currier, EA; Olsson, R; Ma, JN; Burstein, ES; Hacksell, U; Luthman, K Optimization of isochromanone based urotensin II receptor agonists. Bioorg Med Chem18:4844-54 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Urotensin-2 |
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| Name: | Urotensin-2 |
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| Synonyms: | UTS2 | UTS2_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 14297.49 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_643307 |
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| Residue: | 124 |
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| Sequence: | MYKLASCCLLFIGFLNPLLSLPLLDSREISFQLSAPHEDARLTPEELERASLLQILPEML
GAERGDILRKADSSTNIFNPRGNLRKFQDFSGQDPNILLSHLLARIWKPYKKRETPDCFW
KYCV
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| BDBM50416336 |
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| n/a |
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| Name | BDBM50416336 |
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| Synonyms: | CHEMBL380346 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H24ClNO2 |
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| Mol. Mass. | 357.874 |
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| SMILES | CN(C)CCC1(Cc2cc(C)c(C)cc2C(=O)O1)c1ccc(Cl)cc1 |
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| Structure | 
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