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TargetfMet-Leu-Phe receptor 1/2
LigandBDBM50027800
Substrate/Competitorn/a
Meas. Tech.ChEMBL_744776
IC50 2512±n/a nM
Citation Unitt JFagura MPhillips TKing SPerry MMorley AMacDonald CWeaver RChristie JBarber SMohammed RPaul MCook ABaxter A Discovery of small molecule human FPR1 receptor antagonists. Bioorg Med Chem Lett 21:2991-7 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
fMet-Leu-Phe receptor 1/2
Name:fMet-Leu-Phe receptor 1/2
Synonyms:Formyl peptide Receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50027800
n/a
NameBDBM50027800
Synonyms:CHEMBL1770296
TypeSmall organic molecule
Emp. Form.C25H39N3O6S
Mol. Mass.509.659
SMILESCSCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
Structure
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