Reaction Details |
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Target | G-protein coupled receptor 183 |
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Ligand | BDBM50011690 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1351309 (CHEMBL3266158) |
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IC50 | 52±n/a nM |
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Citation | Gessier, F; Preuss, I; Yin, H; Rosenkilde, MM; Laurent, S; Endres, R; Chen, YA; Marsilje, TH; Seuwen, K; Nguyen, DG; Sailer, AW Identification and characterization of small molecule modulators of the Epstein-Barr virus-induced gene 2 (EBI2) receptor. J Med Chem57:3358-68 (2014) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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G-protein coupled receptor 183 |
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Name: | G-protein coupled receptor 183 |
Synonyms: | EBV-induced G-protein coupled receptor 2 | Ebi2 | Epstein-Barr virus-induced G-protein coupled receptor 2 | GP183_MOUSE | Gpr183 |
Type: | PROTEIN |
Mol. Mass.: | 40205.57 |
Organism: | Mus musculus |
Description: | ChEMBL_108312 |
Residue: | 357 |
Sequence: | MANNFTTPLATSHGNNCDLYAHHSTARVLMPLHYSLVFIIGLVGNLLALVVIVQNRKKIN
STTLYSMNLVISDILFTTALPTRIAYYALGFDWRIGDALCRVTALVFYINTYAGVNFMTC
LSIDRFFAVVHPLRYNKIKRIEYAKGVCLSVWILVFAQTLPLLLTPMSKEEGDKTTCMEY
PNFEGTASLPWILLGACLLGYVLPITVILLCYSQICCKLFRTAKQNPLTEKSGVNKKALN
TIILIIVVFILCFTPYHVAIIQHMIKMLCSPGALECGARHSFQISLHFTVCLMNFNCCMD
PFIYFFACKGYKRKVMKMLKRQVSVSISSAVRSAPEENSREMTESQMMIHSKASNGR
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BDBM50011690 |
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n/a |
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Name | BDBM50011690 |
Synonyms: | CHEMBL3262893 |
Type | Small organic molecule |
Emp. Form. | C23H26N2O3 |
Mol. Mass. | 378.4641 |
SMILES | COc1ccc(\C=C\C(=O)N2CCN(CC2)C(=O)c2ccc(C)c(C)c2)cc1 |
Structure |
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