| Reaction Details |
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 | Report a problem with these data |
| Target | Leukotriene B4 receptor 2 |
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| Ligand | BDBM85674 |
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| Substrate/Competitor | n/a |
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| Ki | 3620±n/a nM |
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| Comments | PDSP_1527 |
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| Citation |  Heise, CE; O'Dowd, BF; Figueroa, DJ; Sawyer, N; Nguyen, T; Im, DS; Stocco, R; Bellefeuille, JN; Abramovitz, M; Cheng, R; Williams, DL; Zeng, Z; Liu, Q; Ma, L; Clements, MK; Coulombe, N; Liu, Y; Austin, CP; George, SR; O'Neill, GP; Metters, KM; Lynch, KR; Evans, JF Characterization of the human cysteinyl leukotriene 2 receptor. J Biol Chem275:30531-6 (2000) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Leukotriene B4 receptor 2 |
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| Name: | Leukotriene B4 receptor 2 |
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| Synonyms: | BLT2R | BLTR2 | LT4R2_HUMAN | LTB4 receptor JULF2 | LTB4-R 2 | LTB4-R2 | LTB4R2 | LTB4R2 protein | Leukotriene B4 | Leukotriene B4 R2 | Leukotriene B4 receptor | Leukotriene B4 receptor 2 | Leukotriene B4 receptor BLT2 | Leukotriene b1 | Seven transmembrane receptor BLTR2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 37964.86 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Leukotriene 2 0 HUMAN::Q9NPC1 |
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| Residue: | 358 |
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| Sequence: | MSVCYRPPGNETLLSWKTSRATGTAFLLLAALLGLPGNGFVVWSLAGWRPARGRPLAATL
VLHLALADGAVLLLTPLFVAFLTRQAWPLGQAGCKAVYYVCALSMYASVLLTGLLSLQRC
LAVTRPFLAPRLRSPALARRLLLAVWLAALLLAVPAAVYRHLWRDRVCQLCHPSPVHAAA
HLSLETLTAFVLPFGLMLGCYSVTLARLRGARWGSGRHGARVGRLVSAIVLAFGLLWAPY
HAVNLLQAVAALAPPEGALAKLGGAGQAARAGTTALAFFSSSVNPVLYVFTAGDLLPRAG
PRFLTRLFEGSGEARGGGRSREGTMELRTTPQLKVVGQGRGNGDPGGGMEKDGPEWDL
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| BDBM85674 |
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| n/a |
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| Name | BDBM85674 |
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| Synonyms: | CAS_103177-37-3 | NSC_115100 | Pranlukast |
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| Type | Small organic molecule |
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| Emp. Form. | C27H23N5O4 |
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| Mol. Mass. | 481.5026 |
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| SMILES | O=C(Nc1ccc2c(c1)oc(cc2=O)-c1nnn[nH]1)c1ccc(OCCCCc2ccccc2)cc1 |
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| Structure | 
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