| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM139900 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Binding Assays |
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| Ki | 0.75±n/a nM |
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| Citation |  Frost, JM; Latshaw, SP; Dart, MJ; Carroll, WA; Perez-Medrano, A; Kolasa, T; Patel, MV; Nelson, DW; Li, T; Peddi, S; Wang, X; Liu, B Compounds as cannabinoid receptor ligands US Patent US8895592 Publication Date 11/25/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CNR2_RAT | Cannabinoid CB2 receptor | Cannabinoid receptor | Cnr2 | rCB2 |
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| Type: | Enzyme |
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| Mol. Mass.: | 39366.68 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q9QZN9 |
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| Residue: | 360 |
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| Sequence: | MAGCRELELTNGSNGGLEFNPMKEYMILSDAQQIAVAVLCTLMGLLSALENVAVLYLILS
SQRLRRKPSYLFIGSLAGADFLASVIFACNFVIFHVFHGVDSRNIFLLKIGSVTMTFTAS
VGSLLLTAVDRYLCLCYPPTYKALVTRGRALVALGVMWVLSALISYLPLMGWTCCPSPCS
ELFPLIPNDYLLGWLLFIAILFSGIIYTYGYVLWKAHQHVASLAEHQDRQVPGIARMRLD
VRLAKTLGLVMAVLLICWFPALALMGHSLVTTLSDKVKEAFAFCSMLCLVNSMINPIIYA
LRSGEIRSAAQHCLTGWKKYLQGLGSEGKEEAPKSSVTETEAEVKTTTGPGSRTPGCSNC
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| BDBM139900 |
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| n/a |
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| Name | BDBM139900 |
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| Synonyms: | US8895592, 30 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H28F3N3O2S |
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| Mol. Mass. | 467.548 |
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| SMILES | CC(C)(C)NOc1ccc(cc1C(=O)\N=c1/sc(cn1CCC#C)C(C)(C)C)C(F)(F)F |
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| Structure | 
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