Compile Data Set for Download or QSAR
Found 308 of ki data for polymerid = 188,4952,50007141,520
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM3032(CHEMBL1204168 | CHEMBL29197 | N-(3-bromophenyl)-6,...)copy SMILEScopy InChI
Affinity DataKi:  0.00600nMAssay Description:Inhibition of EGFRChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB82RHPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50238182(CHEMBL4100860)copy SMILEScopy InChI
Affinity DataKi:  0.0700nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98BCKPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Inhibition of wild-type EGFR (unknown origin) by high-throughput biochemical screeningMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged EGFR catalytic domain (669 to 1210 residues) expressed in baculovirus expression system by mass...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50210162(CHEMBL3883534)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Inhibition of PF-06422899 binding to EGFR in human A431 cells after 1 hr by gel-based ABPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125VNCPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613695(CHEMBL5274166)copy SMILES
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50238177(CHEMBL4098072)copy SMILEScopy InChI
Affinity DataKi:  0.350nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin incubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98BCKPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50498973(CHEMBL3734934)copy SMILEScopy InChI
Affinity DataKi: >0.530nMAssay Description:Inhibition of human wild type EGFR using Fl-EEPLYWSFPAKKK-CONH2 as substrate preincubated for 30 mins followed by addition of substrate measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833W1GPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613688(CHEMBL5282716)copy SMILES
Affinity DataKi: <0.600nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613687(CHEMBL5285503)copy SMILES
Affinity DataKi: <0.600nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50141636(CHEMBL3758502)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6MZQPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613684(CHEMBL5280555)copy SMILES
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613695(CHEMBL5274166)copy SMILES
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613698(CHEMBL5282384)copy SMILES
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50141610(CHEMBL3759096)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613699(CHEMBL5279275)copy SMILES
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613686(CHEMBL5276357)copy SMILES
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613695(CHEMBL5274166)copy SMILES
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613699(CHEMBL5279275)copy SMILES
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50141902(CHEMBL3758602)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613699(CHEMBL5279275)copy SMILES
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50238183(CHEMBL4071012)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Inhibition of human N-terminal GST-fused EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus using TK-substrate-biotin incubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98BCKPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50236369((R)-1-morpholino-2-(4-(1-(thiazol-2-ylmethyl)-1H-i...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9H0FPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613693(CHEMBL5281373)copy SMILES
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613687(CHEMBL5285503)copy SMILES
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50112173(CHEMBL3608429)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613698(CHEMBL5282384)copy SMILES
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613698(CHEMBL5282384)copy SMILES
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50450885(CHEMBL4216749)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613685(CHEMBL5273791)copy SMILES
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Centre de Recherches

Curated by ChEMBL
LigandPNGBDBM50236369((R)-1-morpholino-2-(4-(1-(thiazol-2-ylmethyl)-1H-i...)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Inhibition of erbB2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9H0FPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50450884(CHEMBL4211782)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4C0NPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50450887(CHEMBL4211367)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613699(CHEMBL5279275)copy SMILES
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613692(CHEMBL5277269)copy SMILES
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50498976(CHEMBL3736183)copy SMILEScopy InChI
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613699(CHEMBL5279275)copy SMILES
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50450886(CHEMBL4206481)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613695(CHEMBL5274166)copy SMILES
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613693(CHEMBL5281373)copy SMILES
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613698(CHEMBL5282384)copy SMILES
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50237140(CHEMBL4068763)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Reversible inhibition of wild-type human N-terminal GST-tagged EGFR cytoplasmic domain (669 to 1210 end amino acid residues) expressed in baculovirus...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB556RPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613696(CHEMBL5282852)copy SMILES
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50613686(CHEMBL5276357)copy SMILES
Affinity DataKi:  5.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50450871(CHEMBL4205392)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
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