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34 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27690432 75 Discovery of Second Generation Reversible Covalent DPP1 Inhibitors Leading to an Oxazepane Amidoacetonitrile Based Clinical Candidate (AZD7986).EBI Charles River Discovery Research Services
25571794 40 Structure-based design and optimization of potent inhibitors of the adenoviral protease.EBI Novartis Institute For Biomedical Research
24592859 59 Cathepsin C inhibitors: property optimization and identification of a clinical candidate.EBI Astrazeneca
24900293 78 Discovery of novel cyanamide-based inhibitors of cathepsin C.EBI TBA
19715320 87 Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI University of Florida
17535802 91 Inhibition of the activation of multiple serine proteases with a cathepsin C inhibitor requires sustained exposure to prevent pro-enzyme processing.EBI Merck Research Laboratories
18226527 80 The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K.EBI Merck Frosst Centre For Therapeutic Research
19665376 48 Design and synthesis of dipeptidyl nitriles as potent, selective, and reversible inhibitors of cathepsin C.EBI Merck Frosst Canada
19908842 84 Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB.EBI National Human Genome Research Institute
18313933 18 Substrate optimization for monitoring cathepsin C activity in live cells.EBI Genomics Institute of The Novartis Research Foundation
17196818 90 Bicyclic carbamates as inhibitors of papain-like cathepsin proteases.EBI The Genomics Institute of The Novartis Research Foundation
16647256 16 Dipeptidyl nitriles as human dipeptidyl peptidase I inhibitors.EBI Arpida
31145622 91 Identification and Optimization of Novel Cathepsin C Inhibitors Derived from EGFR Inhibitors.EBI National Institute of Biological Sciences (Nibs)
31413809 8 DPP1 Inhibitors: Exploring the Role of Water in the S2 Pocket of DPP1 with Substituted Pyrrolidines.EBI Astrazeneca
3941405 15 Carboxyl-modified amino acids and peptides as protease inhibitors.EBI TBA
23356427 16 Synthesis and carbonic anhydrase inhibitory properties of 1,3-dicarbonyl derivatives of methylaminobenzene-sulfonamide.BDB Sakarya University
2894455 17 Characterization of alpha-2 adrenergic receptors in the OK cell, an opossum kidney cell line.BDB University of Missouri
15710600 29 Demonstration of isoleucine 199 as a structural determinant for the selective inhibition of human monoamine oxidase B by specific reversible inhibitors.BDB Emory University
15225699 27 Preparation of novel aza-1,7-annulated indoles and their conversion to potent indolocarbazole kinase inhibitors.BDB Eli Lilly
 96 Novel Indolocarbazole protein kinase C inhibitors with improved biochemical and physicochemical properties.BDB Tumor Biology Center