The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27504669 |
39 |
Hernandezine, a Bisbenzylisoquinoline Alkaloid with Selective Inhibitory Activity against Multidrug-Resistance-Linked ATP-Binding Cassette Drug Transporter ABCB1. |
Chang Gung Memorial Hospital |
26943020 |
65 |
Pyrrolopyrimidine Derivatives as Novel Inhibitors of Multidrug Resistance-Associated Protein 1 (MRP1, ABCC1). |
University of Bonn |
26774038 |
67 |
Flavonoid derivatives as selective ABCC1 modulators: Synthesis and functional characterization. |
University of Regensburg |
25985195 |
94 |
Potent and Nontoxic Chemosensitizer of P-Glycoprotein-Mediated Multidrug Resistance in Cancer: Synthesis and Evaluation of Methylated Epigallocatechin, Gallocatechin, and Dihydromyricetin Derivatives. |
The Hong Kong Polytechnic University |
21511945 |
7 |
Cannabinoid type 1 receptor antagonists modulate transport activity of multidrug resistance-associated proteins MRP1, MRP2, MRP3, and MRP4. |
Radboud University Nijmegen Medical Centre |
25093931 |
44 |
Trimethoxybenzanilide-based P-glycoprotein modulators: an interesting case of lipophilicity tuning by intramolecular hydrogen bonding. |
Universit£ |
25379609 |
24 |
SAR studies on tetrahydroisoquinoline derivatives: the role of flexibility and bioisosterism to raise potency and selectivity toward P-glycoprotein. |
Universit£ |
25311564 |
30 |
Thieno[2,3-b]pyridines--a new class of multidrug resistance (MDR) modulators. |
Institute of Organic Synthesis |
24184213 |
71 |
Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2). |
University of Bonn |
23851114 |
73 |
Synthesis and biological evaluation of flavones and benzoflavones as inhibitors of BCRP/ABCG2. |
University of Bonn |
23726026 |
12 |
Activity-lipophilicity relationship studies on P-gp ligands designed as simplified tariquidar bulky fragments. |
Universit£ |
23374872 |
27 |
Potent and selective tariquidar bioisosters as potential PET radiotracers for imaging P-gp. |
Universit£ |
23347803 |
29 |
Naphthalenyl derivatives for hitting P-gp/MRP1/BCRP transporters. |
Universit£ |
9188796 |
1 |
Anthracyclines modulate multidrug resistance protein (MRP) mediated organic anion transport. |
Academic Hospital Vrije Universiteit |
8640791 |
1 |
Transport of glutathione, glucuronate, and sulfate conjugates by the MRP gene-encoded conjugate export pump. |
Deutsches Krebsforschungszentrum |
9355767 |
6 |
ATP-dependent transport of bilirubin glucuronides by the multidrug resistance protein MRP1 and its hepatocyte canalicular isoform MRP2. |
Deutsches Krebsforschungszentrum |
11306701 |
5 |
Modulation of multidrug resistance protein 1 (MRP1/ABCC1) transport and atpase activities by interaction with dietary flavonoids. |
Queen'S University |
8621644 |
9 |
ATP-dependent 17 beta-estradiol 17-(beta-D-glucuronide) transport by multidrug resistance protein (MRP). Inhibition by cholestatic steroids. |
Queen'S University |
16434618 |
3 |
Multidrug resistance protein 1 (MRP1, ABCC1) mediates resistance to mitoxantrone via glutathione-dependent drug efflux. |
Wake Forest University School of Medicine |
16384552 |
4 |
Interaction of ivermectin with multidrug resistance proteins (MRP1, 2 and 3). |
Laboratoire De Pharmacologie-Toxicologie Inra |
10612603 |
1 |
Reversal of resistance in multidrug resistance protein (MRP1)-overexpressing cells by LY329146. |
Eli Lilly |
23017888 |
26 |
4-Substituted-2-phenylquinazolines as inhibitors of BCRP. |
University of Bonn |
22366653 |
3 |
Discovery of GS-9451: an acid inhibitor of the hepatitis C virus NS3/4A protease. |
Gilead Sciences |
22165858 |
8 |
Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein. |
Cnrs/Universit£ |
18707884 |
12 |
A 4-aminobenzoic acid derivative as novel lead for selective inhibitors of multidrug resistance-associated proteins. |
University of Bonn |
22112208 |
98 |
Potent galloyl-based selective modulators targeting multidrug resistance associated protein 1 and P-glycoprotein. |
Universit£ |
21530277 |
3 |
Molecular docking studies and in vitro screening of new dihydropyridine derivatives as human MRP1 inhibitors. |
Kakatiya University |
21189339 |
5 |
Interaction potential of etravirine with drug transporters assessed in vitro. |
University Hospital Heidelberg |
21354800 |
77 |
Structure-activity relationships of flavonoids as inhibitors of breast cancer resistance protein (BCRP). |
University of Bonn |
20684594 |
71 |
Phenylsulfonylfuroxans as modulators of multidrug-resistance-associated protein-1 and P-glycoprotein. |
Universita Degli Studi Di Torino |
19932960 |
47 |
Novel lead for potent inhibitors of breast cancer resistance protein (BCRP). |
University of Bonn |
19725578 |
20 |
Modulation of multidrug resistance protein 1 (MRP1/ABCC1)-mediated multidrug resistance by bivalent apigenin homodimers and their derivatives. |
The Hong Kong Polytechnic University |
19580319 |
40 |
Aromatic 2-(thio)ureidocarboxylic acids as a new family of modulators of multidrug resistance-associated protein 1: synthesis, biological evaluation, and structure-activity relationships. |
University of Bonn |
17646169 |
2 |
(R)- and (S)-verapamil differentially modulate the multidrug-resistant protein MRP1. |
Institut De Biologie Et Chimie Des ProtéInes |
16202586 |
7 |
Cyclohexyl-linked tricyclic isoxazoles are potent and selective modulators of the multidrug resistance protein (MRP1). |
Eli Lilly |
16168641 |
35 |
Topological model for the prediction of MRP1 inhibitory activity of pyrrolopyrimidines and templates derived from pyrrolopyrimidine. |
M.D. University |
14998324 |
190 |
Design and synthesis of new templates derived from pyrrolopyrimidine as selective multidrug-resistance-associated protein inhibitors in multidrug resistance. |
Xenova |
14998323 |
79 |
Studies on pyrrolopyrimidines as selective inhibitors of multidrug-resistance-associated protein in multidrug resistance. |
Xenova |
11844674 |
59 |
Studies on quinazolinones as dual inhibitors of Pgp and MRP1 in multidrug resistance. |
Xenova |
32347726 |
41 |
Licochalcone A Selectively Resensitizes ABCG2-Overexpressing Multidrug-Resistant Cancer Cells to Chemotherapeutic Drugs. |
Taipei Chang Gung Memorial Hospital |
27148793 |
112 |
Synthesis and Biological Evaluation of 4-Anilino-quinazolines and -quinolines as Inhibitors of Breast Cancer Resistance Protein (ABCG2). |
University of Bonn |
30594677 |
62 |
Novel chalcone and flavone derivatives as selective and dual inhibitors of the transport proteins ABCB1 and ABCG2. |
Rheinische Friedrich-Wilhelms-University of Bonn |
30584838 |
44 |
Design, Biological Evaluation, and Molecular Modeling of Tetrahydroisoquinoline Derivatives: Discovery of A Potent P-Glycoprotein Ligand Overcoming Multidrug Resistance in Cancer Stem Cells. |
Universit£ |
30947123 |
26 |
Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug resistance (MDR) modulators. |
University of Florence |
31494468 |
61 |
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers. |
University of Florence |
30925062 |
34 |
Identification of Thienopyrimidine Scaffold as an Inhibitor of the ABC Transport Protein ABCC1 (MRP1) and Related Transporters Using a Combined Virtual Screening Approach. |
Rheinische Friedrich-Wilhelms-University of Bonn |
30390439 |
51 |
Synthesis and biological evaluation of quinazoline derivatives - A SAR study of novel inhibitors of ABCG2. |
University of Bonn |
30384046 |
47 |
1,2,3,4-Tetrahydroisoquinoline/2H-chromen-2-one conjugates as nanomolar P-glycoprotein inhibitors: Molecular determinants for affinity and selectivity over multidrug resistance associated protein 1. |
Universit£ |
31465686 |
355 |
Triazole Bridged Flavonoid Dimers as Potent, Nontoxic, and Highly Selective Breast Cancer Resistance Protein (BCRP/ABCG2) Inhibitors. |
Hong Kong Polytechnic University |
17129588 |
30 |
Dibenzocyclooctadiene lignans: a class of novel inhibitors of multidrug resistance-associated protein 1. |
Zhejiang University |
10188979 |
1 |
ATP- and glutathione-dependent transport of chemotherapeutic drugs by the multidrug resistance protein MRP1. |
University Hospital Groningen |
7961706 |
2 |
The MRP gene encodes an ATP-dependent export pump for leukotriene C4 and structurally related conjugates. |
Deutsches Krebsforschungszentrum |
8670053 |
3 |
ATP-dependent glutathione disulphide transport mediated by the MRP gene-encoded conjugate export pump. |
Deutsches Krebsforschungszentrum |
11102445 |
2 |
Glutathione stimulates sulfated estrogen transport by multidrug resistance protein 1. |
Queen'S University |
9647783 |
4 |
Doxorubicin- and daunorubicin-glutathione conjugates, but not unconjugated drugs, competitively inhibit leukotriene C4 transport mediated by MRP/GS-X pump. |
University of Texas M. D. Anderson Cancer Center |
30351934 |
24 |
Discovery of Novel Flavonoid Dimers To Reverse Multidrug Resistance Protein 1 (MRP1, ABCC1) Mediated Drug Resistance in Cancers Using a High Throughput Platform with "Click Chemistry". |
Hong Kong Polytechnic University |
29233614 |
2 |
Monoterpene indole alkaloid azine derivatives as MDR reversal agents. |
Universidade De Lisboa |
28841513 |
117 |
Synthesis and biological investigation of 2,4-substituted quinazolines as highly potent inhibitors of breast cancer resistance protein (ABCG2). |
University of Bonn |
28471656 |
91 |
4-Anilino-2-pyridylquinazolines and -pyrimidines as Highly Potent and Nontoxic Inhibitors of Breast Cancer Resistance Protein (ABCG2). |
University of Bonn |