The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
2153204 |
6 |
Assessment of the in vivo and in vitro opioid activity of bridged hexahydroaporphine and isoquinoline molecules. |
Creighton University |
2709383 |
39 |
Synthesis and pharmacological evaluation of 4,4-disubstituted piperidines. |
Anaquest Pharmaceuticals |
2536439 |
10 |
Synthesis and biological evaluation of 14-alkoxymorphinans. 2. (-)-N-(cyclopropylmethyl)-4,14-dimethoxymorphinan-6-one, a selective mu opioid receptor antagonist. |
University of Innsbruck |
3039139 |
3 |
X-ray crystal structure of the opioid ligand naltrexonazine. |
TBA |
3012085 |
3 |
Probes for narcotic receptor mediated phenomena. 12. cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for delta opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivity. |
TBA |
3009813 |
3 |
Probes for narcotic receptor mediated phenomena. 9. Synthesis of (+/-)-(3 alpha,6a alpha,11a beta)-1,3,4,5,6,11a-hexahydro-2-methyl-2H-3,6a- methanobenzofuro[2,3-c]azocin-10-ol, an oxide-bridged 5-(m-hydroxyphenyl)morphan. |
TBA |
3023609 |
14 |
Probes for narcotic receptor mediated phenomena. 13. Potential irreversible narcotic antagonist-based ligands derived from 6,14-endo-ethenotetrahydronororipavine with 7-(methoxyfumaroyl)amino, (bromoacetyl)amino, or isothiocyanate electrophiles: chemistry, biochemistry, and pharmacology. |
TBA |
2876106 |
6 |
3,7-Diazabicyclane: a new narcotic analgesic. |
TBA |
3020246 |
11 |
Irreversible blockage of opioid receptor types by ester homologues of beta-funaltrexamine. |
TBA |
2863378 |
7 |
Acylmorphinans. A novel class of potent analgesic agents. |
TBA |
2409280 |
35 |
Opioid agonists and antagonists. 6-Desoxy-6-substituted lactone, epoxide, and glycidate ester derivatives of naltrexone and oxymorphone. |
TBA |
2999399 |
4 |
Novel nonnarcotic analgesics with an improved therapeutic ratio. Structure-activity relationships of 8-(methylthio)- and 8-(acylthio)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines. |
TBA |
6094809 |
32 |
Synthesis and biological evaluation of 14-alkoxymorphinans. 1. Highly potent opioid agonists in the series of (-)-14-methoxy-N-methylmorphinan-6-ones. |
TBA |
6315939 |
2 |
14 beta-(2-bromoacetamido)morphine and 14 beta-(2-bromoacetamido)morphinone. |
TBA |
6600791 |
32 |
Synthesis and pharmacological studies of 4,4-disubstituted piperidines: a new class of compounds with potent analgesic properties. |
TBA |
6288945 |
28 |
Potential affinity labels for the opiate receptor based on fentanyl and related compounds. |
TBA |
6276546 |
12 |
Common anionic receptor site hypothesis: its relevance to the antagonist action of naloxone. |
TBA |
6268789 |
22 |
Synthesis of analogues of acetylmethadol and methadol as potential narcotic antagonists. |
TBA |
6268786 |
27 |
Opiate receptor interaction of compounds derived from or structurally related to fentanyl. |
TBA |
6273560 |
16 |
Preparation and analgesic properties of amino acid derivatives of (-)-5,9 alpha-diethyl-2'-hydroxybenzomorphan. |
TBA |
6249930 |
7 |
Synthesis and analgesic activity of some 5-(4-hydroxyphenyl)-2-azabicyclo[3.2.1]octanes. |
TBA |
6248644 |
4 |
Some spiro analogues of the potent analgesic ketobemidone. |
TBA |
2167979 |
43 |
Photoactivatable opiate derivatives as irreversible probes of the mu-opioid receptor. |
Universit£ |
2888899 |
34 |
Combined analgesic/neuroleptic activity in N-butyrophenone prodine-like compounds. |
Istituto Superiore Di Sanit£ |
3007760 |
93 |
N-substituent modulation of opiate agonist/antagonist activity in resolved 3-methyl-3-(m-hydroxyphenyl)piperidines. |
TBA |
8411007 |
392 |
Chemistry, binding affinities, and behavioral properties of a new class of"antineophobic" mitochondrial DBI receptor complex (mDRC) ligands. |
Mayo Foundation |
6313921 |
10 |
Synthesis and pharmacological characterization of (+/-)-5,9 alpha-dimethyl-2-[2-(4-fluorophenyl)ethyl]-2'-hydroxy-6,7-benzomorphan (fluorophen), a ligand suitable for visualization of opiate receptors in vivo. |
TBA |
3746815 |
15 |
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin. |
TBA |
2153212 |
87 |
Cholecystokinin-A receptor ligands based on the kappa-opioid agonist tifluadom. |
Merck Sharp & Dohme Research Laboratories |
1323682 |
61 |
Novel indolodioxanes with antihypertensive effects: potent ligands for the 5-HT1A receptor. |
Upjohn |