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32 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
2153204 6 Assessment of the in vivo and in vitro opioid activity of bridged hexahydroaporphine and isoquinoline molecules.EBI Creighton University
2709383 39 Synthesis and pharmacological evaluation of 4,4-disubstituted piperidines.EBI Anaquest Pharmaceuticals
2536439 10 Synthesis and biological evaluation of 14-alkoxymorphinans. 2. (-)-N-(cyclopropylmethyl)-4,14-dimethoxymorphinan-6-one, a selective mu opioid receptor antagonist.EBI University of Innsbruck
3039139 3 X-ray crystal structure of the opioid ligand naltrexonazine.EBI TBA
3012085 3 Probes for narcotic receptor mediated phenomena. 12. cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for delta opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivity.EBI TBA
3009813 3 Probes for narcotic receptor mediated phenomena. 9. Synthesis of (+/-)-(3 alpha,6a alpha,11a beta)-1,3,4,5,6,11a-hexahydro-2-methyl-2H-3,6a- methanobenzofuro[2,3-c]azocin-10-ol, an oxide-bridged 5-(m-hydroxyphenyl)morphan.EBI TBA
3023609 14 Probes for narcotic receptor mediated phenomena. 13. Potential irreversible narcotic antagonist-based ligands derived from 6,14-endo-ethenotetrahydronororipavine with 7-(methoxyfumaroyl)amino, (bromoacetyl)amino, or isothiocyanate electrophiles: chemistry, biochemistry, and pharmacology.EBI TBA
2876106 6 3,7-Diazabicyclane: a new narcotic analgesic.EBI TBA
3020246 11 Irreversible blockage of opioid receptor types by ester homologues of beta-funaltrexamine.EBI TBA
2863378 7 Acylmorphinans. A novel class of potent analgesic agents.EBI TBA
2409280 35 Opioid agonists and antagonists. 6-Desoxy-6-substituted lactone, epoxide, and glycidate ester derivatives of naltrexone and oxymorphone.EBI TBA
2999399 4 Novel nonnarcotic analgesics with an improved therapeutic ratio. Structure-activity relationships of 8-(methylthio)- and 8-(acylthio)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines.EBI TBA
6094809 32 Synthesis and biological evaluation of 14-alkoxymorphinans. 1. Highly potent opioid agonists in the series of (-)-14-methoxy-N-methylmorphinan-6-ones.EBI TBA
6315939 2 14 beta-(2-bromoacetamido)morphine and 14 beta-(2-bromoacetamido)morphinone.EBI TBA
6600791 32 Synthesis and pharmacological studies of 4,4-disubstituted piperidines: a new class of compounds with potent analgesic properties.EBI TBA
6288945 28 Potential affinity labels for the opiate receptor based on fentanyl and related compounds.EBI TBA
6276546 12 Common anionic receptor site hypothesis: its relevance to the antagonist action of naloxone.EBI TBA
6268789 22 Synthesis of analogues of acetylmethadol and methadol as potential narcotic antagonists.EBI TBA
6268786 27 Opiate receptor interaction of compounds derived from or structurally related to fentanyl.EBI TBA
6273560 16 Preparation and analgesic properties of amino acid derivatives of (-)-5,9 alpha-diethyl-2'-hydroxybenzomorphan.EBI TBA
6249930 7 Synthesis and analgesic activity of some 5-(4-hydroxyphenyl)-2-azabicyclo[3.2.1]octanes.EBI TBA
6248644 4 Some spiro analogues of the potent analgesic ketobemidone.EBI TBA
2167979 43 Photoactivatable opiate derivatives as irreversible probes of the mu-opioid receptor.EBI Universit£
2888899 34 Combined analgesic/neuroleptic activity in N-butyrophenone prodine-like compounds.EBI Istituto Superiore Di Sanit£
3007760 93 N-substituent modulation of opiate agonist/antagonist activity in resolved 3-methyl-3-(m-hydroxyphenyl)piperidines.EBI TBA
8411007 392 Chemistry, binding affinities, and behavioral properties of a new class of"antineophobic" mitochondrial DBI receptor complex (mDRC) ligands.EBI Mayo Foundation
6313921 10 Synthesis and pharmacological characterization of (+/-)-5,9 alpha-dimethyl-2-[2-(4-fluorophenyl)ethyl]-2'-hydroxy-6,7-benzomorphan (fluorophen), a ligand suitable for visualization of opiate receptors in vivo.EBI TBA
3746815 15 In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.EBI TBA
2153212 87 Cholecystokinin-A receptor ligands based on the kappa-opioid agonist tifluadom.EBI Merck Sharp & Dohme Research Laboratories
1323682 61 Novel indolodioxanes with antihypertensive effects: potent ligands for the 5-HT1A receptor.EBI Upjohn