The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
25470070 |
81 |
Probing the carboxyester side chain in controlled deactivation (-)-d(8)-tetrahydrocannabinols. |
Northeastern University |
28085283 |
118 |
Design, Synthesis, and Biological Evaluation of Novel, Non-Brain-Penetrant, Hybrid Cannabinoid CB |
National Institute On Alcohol Abuse and Alcoholism |
8411021 |
3 |
Two new unsaturated fatty acid ethanolamides in brain that bind to the cannabinoid receptor. |
Hebrew University |
27240274 |
37 |
A critical review of both the synthesis approach and the receptor profile of the 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide and analogue derivatives. |
Neuroscienze Pharmaness S.C.A R.L. |
26275680 |
68 |
Synthesis and biological evaluation of (3',5'-dichloro-2,6-dihydroxy-biphenyl-4-yl)-aryl/alkyl-methanone selective CB2 inverse agonist. |
University of Tennessee Health Science Center |
25950914 |
84 |
Discovery of a high affinity and selective pyridine analog as a potential positron emission tomography imaging agent for cannabinoid type 2 receptor. |
Institute of Pharmaceutical Sciences |
25760146 |
49 |
3'-functionalized adamantyl cannabinoid receptor probes. |
University of Hawaii At Manoa |
25701254 |
48 |
Novel tail and head group prostamide probes. |
Northeastern University |
25134064 |
40 |
Tricyclic pyrazoles part 7. Discovery of potent and selective dihydrothienocyclopentapyrazole derived CB2 ligands. |
Universit£ |
25488844 |
154 |
Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists. |
Arena Pharmaceuticals |
24922543 |
24 |
Tricyclic pyrazoles. Part 6. Benzofuro[3,2-c]pyrazole: a versatile architecture for CB2 selective ligands. |
Universit£ |
24900848 |
11 |
C-ring cannabinoid lactones: a novel cannabinergic chemotype. |
Northeastern University |
23865723 |
169 |
Therapeutic utility of cannabinoid receptor type 2 (CB(2)) selective agonists. |
Arena Pharmaceuticals |
23621789 |
69 |
Novel adamantyl cannabinoids as CB1 receptor probes. |
Northeastern University |
23380378 |
127 |
Highly potent and selective cannabinoid receptor 2 agonists: initial hit optimization of an adamantyl hit series identified from high-through-put screening. |
F. Hoffmann-La Roche |
23357307 |
14 |
Novel pyrazole derivatives as neutral CB1 antagonists with significant activity towards food intake. |
Neuroscienze Pharmaness S.C.A R.L. |
23147076 |
163 |
Structure-activity relationships of 2-arylamido-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxamide derivatives as cannabinoid receptor agonists and their analgesic action. |
Nycomed Pharma |
23083016 |
20 |
Sulfonyl fluoride inhibitors of fatty acid amide hydrolase. |
Northeastern University |
22738638 |
59 |
Assay and inhibition of diacylglycerol lipase activity. |
Northeastern University |
22796181 |
51 |
C3-heteroaroyl cannabinoids as photolabeling ligands for the CB2 cannabinoid receptor. |
University of Hawaii At Manoa |
17149879 |
40 |
Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide. |
Universit£ |
17004710 |
51 |
Design, synthesis, and biological evaluation of new 1,8-naphthyridin-4(1H)-on-3-carboxamide and quinolin-4(1H)-on-3-carboxamide derivatives as CB2 selective agonists. |
Universit£ |
16190764 |
24 |
Potent cannabinergic indole analogues as radioiodinatable brain imaging agents for the CB1 cannabinoid receptor. |
Northeastern University |
8809166 |
10 |
Unsaturated side chain beta-11-hydroxyhexahydrocannabinol analogs. |
University of Hawaii |
21880487 |
21 |
Conformationally constrained analogs of BAY 59-3074 as novel cannabinoid receptor ligands. |
Northeastern University |
20925434 |
43 |
Novel 1',1'-chain substituted hexahydrocannabinols: 9ß-hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a highly potent cannabinoid receptor 1 (CB1) agonist. |
Northeastern University |
20593789 |
47 |
Heteroadamantyl cannabinoids. |
University of Hawaii At Manoa |
20591666 |
66 |
A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase. |
Università |
18826296 |
12 |
Bornyl- and isobornyl-Delta8-tetrahydrocannabinols: a novel class of cannabinergic ligands. |
Northeastern University |
18723350 |
37 |
Development of novel tail-modified anandamide analogs. |
Northeastern University |
18038967 |
12 |
Cannabilactones: a novel class of CB2 selective agonists with peripheral analgesic activity. |
Northeastern University |
17826996 |
5 |
Conformationally constrained analogues of 2-arachidonoylglycerol. |
Northeastern University |
17672444 |
22 |
C1'-cycloalkyl side chain pharmacophore in tetrahydrocannabinols. |
National Hellenic Research Foundation |
17531479 |
65 |
2-Arylimino-5,6-dihydro-4H-1,3-thiazines as a new class of cannabinoid receptor agonists. Part 2: orally bioavailable compounds. |
Shionogi |
17521907 |
50 |
2-Arylimino-5,6-dihydro-4H-1,3-thiazines as a new class of cannabinoid receptor agonists. Part 1: discovery of CB2 receptor selective compounds. |
Shionogi |
16387492 |
26 |
Structural modifications of the cannabinoid side chain towards C3-aryl and 1',1'-cycloalkyl-1'-cyano cannabinoids. |
National Hellenic Research Foundation |
16279795 |
36 |
Tricyclic pyrazoles. 3. Synthesis, biological evaluation, and molecular modeling of analogues of the cannabinoid antagonist 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide. |
Università |
15999995 |
12 |
Adamantyl cannabinoids: a novel class of cannabinergic ligands. |
Northeastern University |
12852753 |
17 |
Pharmacophoric requirements for the cannabinoid side chain. Probing the cannabinoid receptor subsite at C1'. |
National Hellenic Research Foundation |
12443781 |
22 |
Novel 1',1'-chain substituted Delta(8)-tetrahydrocannabinols. |
National Hellenic Research Foundation |
27624523 |
33 |
Synthesis, molecular modeling and SAR study of novel pyrazolo[5,1-f][1,6]naphthyridines as CB |
Universit£ |
27367336 |
78 |
Novel C-Ring-Hydroxy-Substituted Controlled Deactivation Cannabinergic Analogues. |
Northeastern University |
30816712 |
78 |
Plant-Based Modulators of Endocannabinoid Signaling. |
Concordia University Wisconsin |
10465529 |
9 |
Novel conformationally restricted tetracyclic analogs of delta8-tetrahydrocannabinol. |
University of Connecticut |
10052983 |
40 |
Structure-activity relationships of pyrazole derivatives as cannabinoid receptor antagonists. |
University of Connecticut |
9876105 |
75 |
Novel analogues of arachidonylethanolamide (anandamide): affinities for the CB1 and CB2 cannabinoid receptors and metabolic stability. |
University of Connecticut |
29939744 |
179 |
Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure-Functional Selectivity Relationships (SFSRs) and Therapeutic Potential. |
Shanghaitech University |
9733485 |
16 |
Classical/nonclassical hybrid cannabinoids: southern aliphatic chain-functionalized C-6beta methyl, ethyl, and propyl analogues. |
University of Hawaii |
9544219 |
12 |
Pharmacophoric requirements for cannabinoid side chains: multiple bond and C1'-substituted delta 8-tetrahydrocannabinols. |
National Hellenic Research Foundation |
8893848 |
21 |
Head group analogs of arachidonylethanolamide, the endogenous cannabinoid ligand. |
University of Connecticut |
24286207 |
30 |
Controlled-deactivation cannabinergic ligands. |
Northeastern University |
24095014 |
52 |
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors. |
Uos of Cagliari |
16190768 |
6 |
High affinity electrophilic and photoactivatable covalent endocannabinoid probes for the CB1 receptor. |
Northeastern University |
30122284 |
70 |
Oximes short-acting CB1 receptor agonists. |
Northeastern University |
30196704 |
90 |
( R)- N-(1-Methyl-2-hydroxyethyl)-13-( S)-methyl-arachidonamide (AMG315): A Novel Chiral Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes. |
Northeastern University |
28792219 |
61 |
Novel Diarylurea Based Allosteric Modulators of the Cannabinoid CB1 Receptor: Evaluation of Importance of 6-Pyrrolidinylpyridinyl Substitution. |
Research Triangle Institute |
26575582 |
15 |
Development of 2-(Substituted Benzylamino)-4-Methyl-1, 3-Thiazole-5-Carboxylic Acid Derivatives as Xanthine Oxidase Inhibitors and Free Radical Scavengers. |
Jamia Hamdard |