The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26288216 |
579 |
Pharmaceutical Optimization of Peptide Toxins for Ion Channel Targets: Potent, Selective, and Long-Lived Antagonists of Kv1.3. |
Amgen |
23084278 |
21 |
Structure-activity relationship exploration of Kv1.3 blockers based on diphenoxylate. |
Monash University (Parkville Campus) |
18289849 |
8 |
Synthesis and biological evaluation of chalcones as inhibitors of the voltage-gated potassium channel Kv1.3. |
The Walter and Eliza Hall Institute of Medical Research |
11356099 |
20 |
Recent developments in the biology and medicinal chemistry of potassium channel modulators: update from a decade of progress. |
Abbott Laboratories |
20974533 |
99 |
Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 ion channel blockers. Part 2. |
Glaxosmithkline |
20971642 |
59 |
N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 inhibitors. Part 1. |
Glaxosmithkline |
19888755 |
43 |
Selective Kv1.5 blockers: development of (R)-1-(methylsulfonylamino)-3-[2-(4-methoxyphenyl)ethyl]-4-(4-methoxyphenyl)-2-imidazolidinone (KVI-020/WYE-160020) as a potential treatment for atrial arrhythmia. |
Wyeth Research |
19056148 |
27 |
4-Phenoxybutoxy-substituted heterocycles--a structure-activity relationship study of blockers of the lymphocyte potassium channel Kv1.3. |
University of California |
| 1 |
The SAR of UK-78,282: A novel blocker of human T cell Kv1.3 potassium channels |
TBA |
19282171 |
29 |
Inhibitors of potassium channels KV1.3 and IK-1 as immunosuppressants. |
4Sc |
19042133 |
4 |
Gamma-pyrone natural products--a privileged compound class provided by nature. |
Institute of Molecular Physiology |
15603971 |
63 |
Potent Kv1.3 inhibitors from correolide-modification of the C18 position. |
Merck Research Laboratories |
15084131 |
27 |
Khellinone derivatives as blockers of the voltage-gated potassium channel Kv1.3: synthesis and immunosuppressive activity. |
Institute of Medical Research Biotechnology Centre |
12643934 |
109 |
Benzamide derivatives as blockers of Kv1.3 ion channel. |
Merck Research Laboratories |
12570371 |
33 |
Identification, synthesis, and activity of novel blockers of the voltage-gated potassium channel Kv1.5. |
Aventis Pharma Deutschland |
10612582 |
13 |
Blockers of human T cell Kv1.3 potassium channels using de novo ligand design and solid-phase parallel combinatorial chemistry. |
University of California |
7540207 |
56 |
Novel inhibitors of potassium ion channels on human T lymphocytes. |
Sanofi Winthrop |
28802123 |
89 |
Clathrodin, hymenidin and oroidin, and their synthetic analogues as inhibitors of the voltage-gated potassium channels. |
University of Ljubljana |