Found 79 hits for monomerid = 30707 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PCBioAssay
| n/a | n/a | n/a | n/a | 197 | n/a | n/a | 7.4 | 23 |
The Scripps Research Institute Molecular Screening Center
Curated by PubChem BioAssay
| Assay Description A cell line containing the human 5-HT1a receptor, the promiscuous G-alpha-15 protein (Ga15) as well as the beta-lactamase (BLA) reporter-gene under c... |
PubChem Bioassay (2007)
BindingDB Entry DOI: 10.7270/Q2WW7G03 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| | 70 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
Virginia Commonwealth University
| Assay Description The h5-HT6 radioligand binding assays were performed as previously described. In brief, h5-HT6 cDNA was transiently expressed in HEK-293 cells using... |
Medicinal Chemistry Research 14: 1-18 (2005)
BindingDB Entry DOI: 10.7270/Q2NG4P78 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
UniProtKB/SwissProt
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| PCBioAssay
| n/a | n/a | n/a | n/a | 1.06E+3 | n/a | n/a | 7.4 | 23 |
The Scripps Research Institute Molecular Screening Center
Curated by PubChem BioAssay
| Assay Description A cell line containing the human 5-HT1a receptor, the promiscuous G-alpha-15 protein (Ga15) as well as the beta-lactamase (BLA) reporter-gene under c... |
PubChem Bioassay (2007)
BindingDB Entry DOI: 10.7270/Q21N7ZG0 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1E
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| PCBioAssay
| n/a | n/a | n/a | n/a | 92 | n/a | n/a | 7.4 | 23 |
The Scripps Research Institute Molecular Screening Center
Curated by PubChem BioAssay
| Assay Description The CHO cell line was cultured in T-175 sq cm Corning flasks (part 431080) at 37 deg C and 95% RH. The HTS assay began by dispensing 10 microliters o... |
PubChem Bioassay (2007)
BindingDB Entry DOI: 10.7270/Q2Q52MZM |
More data for this Ligand-Target Pair | |
Sphingosine 1-phosphate receptor 3
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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| PCBioAssay
| n/a | n/a | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center
Curated by PubChem BioAssay
| Assay Description External Assay ID: S1P3_EC50_CS_5HT1e_Agonist Name: S1P3 Dose Response Assay Counterscreen for 5-Hydroxytryptamine(Serotonin) Receptor Subtype 1E ... |
PubChem Bioassay (2007)
BindingDB Entry DOI: 10.7270/Q2PN941W |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1E
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| PubMed
| 528 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation
Curated by PDSP Ki Database
| |
Mol Pharmacol 42: 180-5 (1992)
BindingDB Entry DOI: 10.7270/Q2416VJ0 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
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| Article PubMed
| 39.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM U. 114
Curated by PDSP Ki Database
| |
Nature 305: 140-2 (1983)
Article DOI: 10.1038/305140a0 BindingDB Entry DOI: 10.7270/Q2S46QFX |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
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| Article PubMed
| 288 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM U. 114
Curated by PDSP Ki Database
| |
Nature 305: 140-2 (1983)
Article DOI: 10.1038/305140a0 BindingDB Entry DOI: 10.7270/Q2S46QFX |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| PubMed
| 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Stanford University
Curated by PDSP Ki Database
| |
J Neurosci 9: 3482-90 (1989)
BindingDB Entry DOI: 10.7270/Q2FX77Z2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2B
(BOVINE) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway
UniProtKB/TrEMBL
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| PubMed
| 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Stanford University
Curated by PDSP Ki Database
| |
J Neurosci 9: 3482-90 (1989)
BindingDB Entry DOI: 10.7270/Q2FX77Z2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(GUINEA PIG) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
UniProtKB/SwissProt
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| Article PubMed
| 107 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Syntex Discovery Research
Curated by PDSP Ki Database
| |
Br J Pharmacol 115: 107-16 (1995)
Article DOI: 10.1111/j.1476-5381.1995.tb16327.x BindingDB Entry DOI: 10.7270/Q2610XTR |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(GUINEA PIG) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
UniProtKB/SwissProt
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| Article PubMed
| 13.2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Syntex Discovery Research
Curated by PDSP Ki Database
| |
Br J Pharmacol 115: 107-16 (1995)
Article DOI: 10.1111/j.1476-5381.1995.tb16327.x BindingDB Entry DOI: 10.7270/Q2610XTR |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(RAT) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway
UniProtKB/SwissProt
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| PubMed
| 79.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Neurological Disorders and Stroke
Curated by PDSP Ki Database
| |
Mol Pharmacol 43: 320-7 (1993)
BindingDB Entry DOI: 10.7270/Q2ST7NCG |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| Article PubMed
| 23.4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1D
(Dog) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
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| Article PubMed
| 5.12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1E
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| Article PubMed
| 525 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1F
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| Article PubMed
| 37.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(RAT) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway
UniProtKB/SwissProt
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| Article PubMed
| 79.4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| Article PubMed
| 20.9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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Patents
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| Article PubMed
| 8.31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Alberta
Curated by PDSP Ki Database
| |
Neuropharmacology 33: 275-317 (1994)
Article DOI: 10.1016/0028-3908(94)90059-0 BindingDB Entry DOI: 10.7270/Q2M043X2 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1F
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| Article PubMed
| 37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation
Curated by PDSP Ki Database
| |
Proc Natl Acad Sci U S A 90: 408-12 (1993)
Article DOI: 10.1073/pnas.90.2.408 BindingDB Entry DOI: 10.7270/Q2862DZF |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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Patents
Similars
| PubMed
| 20.9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Neurological Disorders and Stroke
Curated by PDSP Ki Database
| |
J Biol Chem 268: 18200-4 (1993)
BindingDB Entry DOI: 10.7270/Q2V1239R |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 7
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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Patents
Similars
| PubMed
| 8.26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Neurological Disorders and Stroke
Curated by PDSP Ki Database
| |
J Biol Chem 268: 18200-4 (1993)
BindingDB Entry DOI: 10.7270/Q2V1239R |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| Article PubMed
| 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Albany Medical College
Curated by PDSP Ki Database
| |
Synapse 35: 144-50 (2000)
Article DOI: 10.1002/(SICI)1098-2396(200002)35:2<144::AID-SYN7>3.0.CO;2-K BindingDB Entry DOI: 10.7270/Q2ST7NDX |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| Article PubMed
| 1.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Albany Medical College
Curated by PDSP Ki Database
| |
Synapse 35: 144-50 (2000)
Article DOI: 10.1002/(SICI)1098-2396(200002)35:2<144::AID-SYN7>3.0.CO;2-K BindingDB Entry DOI: 10.7270/Q2ST7NDX |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| PubMed
| 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description Affinity of the compound on 5-hydroxytryptamine 1A receptor labeled by [3H]-8-OH-DPAT |
J Med Chem 35: 2061-4 (1992)
BindingDB Entry DOI: 10.7270/Q2PG1QN7 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| PubMed
| n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc.
Curated by ChEMBL
| Assay Description Compound was evaluated for binding affinity towards 5-hydroxytryptamine 1D receptor in bovine caudate using [3H]- serotonin as radioligand |
J Med Chem 35: 3625-32 (1992)
BindingDB Entry DOI: 10.7270/Q2125RK7 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
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| PubMed
| n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc.
Curated by ChEMBL
| Assay Description Compound was evaluated for binding affinity towards 5-hydroxytryptamine 1A receptor in rat cortex using [3H]-8-OH-DPAT as radioligand |
J Med Chem 35: 3625-32 (1992)
BindingDB Entry DOI: 10.7270/Q2125RK7 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc.
Curated by ChEMBL
| Assay Description Binding affinity of the compound towards 5-hydroxytryptamine 1C receptor using [3H]-mesulergine as radioligand |
J Med Chem 35: 3625-32 (1992)
BindingDB Entry DOI: 10.7270/Q2125RK7 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PubMed
| n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc
Curated by ChEMBL
| Assay Description Binding affinity of the compound against 5-hydroxytryptamine 1A receptor |
J Med Chem 35: 4503-5 (1992)
BindingDB Entry DOI: 10.7270/Q29C6WC5 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
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| PubMed
| n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc
Curated by ChEMBL
| Assay Description Binding affinity of the compound against 5-hydroxytryptamine 1C receptor |
J Med Chem 35: 4503-5 (1992)
BindingDB Entry DOI: 10.7270/Q29C6WC5 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| PubMed
| n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc
Curated by ChEMBL
| Assay Description Binding affinity of the compound against 5-hydroxytryptamine 1B receptor |
J Med Chem 35: 4503-5 (1992)
BindingDB Entry DOI: 10.7270/Q29C6WC5 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1D
(GUINEA PIG) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
UniProtKB/SwissProt
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| PubMed
| n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc
Curated by ChEMBL
| Assay Description Binding affinity of the compound against 5-hydroxytryptamine 1D receptor |
J Med Chem 35: 4503-5 (1992)
BindingDB Entry DOI: 10.7270/Q29C6WC5 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1B
(Rattus norvegicus (Rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| PubMed
| 350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Evaluated for binding affinity towards 5-hydroxytryptamine 1B receptor |
J Med Chem 31: 867-70 (1988)
BindingDB Entry DOI: 10.7270/Q2QN65SB |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
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| PubMed
| 7.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity towards 5-hydroxytryptamine 1A receptor |
J Med Chem 31: 867-70 (1988)
BindingDB Entry DOI: 10.7270/Q2QN65SB |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity of compound towards 5-hydroxytryptamine 1A receptor in rat striatal membranes by [3H]-OH-DPAT displacement. |
J Med Chem 32: 1921-6 (1989)
BindingDB Entry DOI: 10.7270/Q2J67FWB |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| PubMed
| 620 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Affinity against 5-hydroxytryptamine 2A receptor (K) labeled with [3H]-ketanserin. |
J Med Chem 37: 1929-35 (1994)
BindingDB Entry DOI: 10.7270/Q2GQ6WT0 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| 960 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Affinity against 5-hydroxytryptamine 2C receptor in J1 cells transfected with the rat 5-HT2C gene labeled with [3H]-mesulergine. |
J Med Chem 37: 1929-35 (1994)
BindingDB Entry DOI: 10.7270/Q2GQ6WT0 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Affinity against 5-hydroxytryptamine 2A receptor (D) labeled with [125I]-DOI. |
J Med Chem 37: 1929-35 (1994)
BindingDB Entry DOI: 10.7270/Q2GQ6WT0 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
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| Article PubMed
| 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity of the compound towards 5-hydroxytryptamine 1D receptor was determined in calf striatum homogenate |
J Med Chem 39: 314-22 (1996)
Article DOI: 10.1021/jm950498t BindingDB Entry DOI: 10.7270/Q2DJ5DRK |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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CHEMBL KEGG PC cid PC sid UniChem
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Similars
| Article PubMed
| n/a | n/a | 9.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Inhibition of [125I]DOI binding to 5HT2A receptor in rat cerebral cortex |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue University
Curated by ChEMBL
| Assay Description Compound was tested for binding affinity using [3H]-MDL-100,907 at 5-hydroxytryptamine 2A receptor sites in rat cortical homogenate. |
J Med Chem 42: 4257-63 (1999)
BindingDB Entry DOI: 10.7270/Q2FX78PW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity for human 5-hydroxytryptamine 6 receptor expressed in HEK 293 human embryonic kidney cells, [3H]-lysergic acid diethylamide as radio... |
J Med Chem 43: 1011-8 (2000)
BindingDB Entry DOI: 10.7270/Q2CF9PBP |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 6
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| PubMed
| 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University
Curated by ChEMBL
| Assay Description Binding affinity against human 5-hydroxytryptamine 6 receptor stably transfected to HEK 293 human embryonic kidney cells using [3H]-lysergic acid die... |
Bioorg Med Chem Lett 10: 2295-9 (2001)
BindingDB Entry DOI: 10.7270/Q29C6WP6 |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cells |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 462 | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Activity against 5HT2A mediated intracellular calcium mobilization by FLIPR in rat vascular smooth muscle cells |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2B
(RAT) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 240 | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Activity against 5HT2B receptor in longitudinal stomach fundus strips in wistar rats |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | n/a | n/a | 78 | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Activity against recombinant rat 5HT2C mediated intracellular calcium mobilization by FLIPR in SR3T3 cells |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cells |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human)) | BDBM30707
![PNG](/data/jpeg/tenK3/BindingDB_30707.png) (2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamin...)Show InChI InChI=1S/C13H18N2O/c1-15(2)7-6-10-9-14-13-5-4-11(16-3)8-12(10)13/h4-5,8-9,14H,6-7H2,1-3H3 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
CHEMBL KEGG PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 52 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alcon Research, Ltd.
Curated by ChEMBL
| Assay Description Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cells |
J Med Chem 49: 318-28 (2006)
Article DOI: 10.1021/jm050663x BindingDB Entry DOI: 10.7270/Q23B5ZQW |
More data for this Ligand-Target Pair | |