Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82310![]() (Purine, 5) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | 4.30E+3 | -31.9 | 1.02E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286099![]() (N-(5-(ethylsulfonyl)-5-azaspiro[2.4]heptan-7-yl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286098![]() ((R)-3-((7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286095![]() ((R)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase, cytoplasmic (Homo sapiens (Human)) | BDBM50458119![]() (Leusa) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid PDB UniChem | PDB PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of catalytic activity of LRS (unknown origin) by aminoleucylation assay | Citation and Details BindingDB Entry DOI: 10.7270/Q2QR51RW | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Non-receptor tyrosine-protein kinase TYK2 (Homo sapiens (Human)) | BDBM286098![]() ((R)-3-((7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 24.7 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286096![]() (3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 29.3 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Non-receptor tyrosine-protein kinase TYK2 (Homo sapiens (Human)) | BDBM286096![]() (3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 40.4 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286098![]() ((R)-3-((7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 58.6 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase, cytoplasmic (Homo sapiens (Human)) | BDBM50550346![]() (CHEMBL4558130) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of catalytic activity of LRS (unknown origin) by aminoleucylation assay | Citation and Details BindingDB Entry DOI: 10.7270/Q2QR51RW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK3 (Homo sapiens (Human)) | BDBM286098![]() ((R)-3-((7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286096![]() (3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 148 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Non-receptor tyrosine-protein kinase TYK2 (Homo sapiens (Human)) | BDBM286099![]() (N-(5-(ethylsulfonyl)-5-azaspiro[2.4]heptan-7-yl)-N...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 198 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Non-receptor tyrosine-protein kinase TYK2 (Homo sapiens (Human)) | BDBM286095![]() ((R)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 252 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leucine--tRNA ligase, cytoplasmic (Homo sapiens (Human)) | BDBM50550345![]() (CHEMBL4104169) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | PubMed | n/a | n/a | 337 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of catalytic activity of LRS (unknown origin) by aminoleucylation assay | Citation and Details BindingDB Entry DOI: 10.7270/Q2QR51RW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286095![]() ((R)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 412 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286099![]() (N-(5-(ethylsulfonyl)-5-azaspiro[2.4]heptan-7-yl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 422 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK3 (Homo sapiens (Human)) | BDBM286096![]() (3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 694 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286097![]() ((S)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 787 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK3 (Homo sapiens (Human)) | BDBM286097![]() ((S)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK3 (Homo sapiens (Human)) | BDBM286099![]() (N-(5-(ethylsulfonyl)-5-azaspiro[2.4]heptan-7-yl)-N...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Non-receptor tyrosine-protein kinase TYK2 (Homo sapiens (Human)) | BDBM286097![]() ((S)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK1 (Homo sapiens (Human)) | BDBM286097![]() ((S)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase JAK3 (Homo sapiens (Human)) | BDBM286095![]() ((R)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
YANG JI CHEMICAL CO., LTD.; HAN WHA PHARMA CO., LTD. US Patent | Assay Description Kinases used were human-derived JAK1, JAK2, JAK3, and TYK2 (Millipore, Germany). Each of these kinases was diluted with a suitable buffer solution as... | US Patent US10081635 (2018) BindingDB Entry DOI: 10.7270/Q2R213D4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473488![]() (CHEMBL141477) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473487![]() (CHEMBL336919) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473496![]() (CHEMBL136246) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473495![]() (CHEMBL139282) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473493![]() (CHEMBL138292) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473490![]() (CHEMBL139200) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473494![]() (Myoseverin) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82329![]() (Purine, 24) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.27E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82307![]() (Purine, 2) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.35E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82308![]() (Purine, 3) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.37E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82322![]() (Purine, 17) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.82E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82328![]() (Purine, 23) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82324![]() (Purine, 19) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.34E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473492![]() (CHEMBL140654) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473489![]() (CHEMBL140649) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82327![]() (Purine, 22) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82326![]() (Purine, 21) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.88E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82309![]() (Purine, 4) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.34E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82325![]() (Purine, 20) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.90E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Similar to alpha-tubulin isoform 1 (Bos taurus) | BDBM50473491![]() (CHEMBL343349) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
New York University Curated by ChEMBL | Assay Description Inhibition of tubulin polymerization using bovine brain tubulin | J Med Chem 44: 4497-500 (2001) Article DOI: 10.1021/jm010451+ BindingDB Entry DOI: 10.7270/Q2XW4NJH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82306![]() (Purine, 1) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.71E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82318![]() (Purine, 13) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82323![]() (Purine, 18) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.76E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82313![]() (Purine, 8) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.02E+5 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82320![]() (Purine, 15) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.17E+5 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inositol-trisphosphate 3-kinase A (Homo sapiens (Human)) | BDBM82312![]() (Purine, 7) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.38E+5 | n/a | n/a | n/a | n/a | 8.0 | 37 |
New York University | Assay Description IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and... | Chembiochem 3: 897-901 (2002) Article DOI: 10.1002/1439-7633(20020902)3:9 BindingDB Entry DOI: 10.7270/Q2DJ5D4H | |||||||||||
More data for this Ligand-Target Pair |
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