Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413761![]() (CHEMBL390094) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Salerno Curated by ChEMBL | Assay Description Binding affinity towards human Urotensin 2 receptor was determined | J Med Chem 47: 1652-61 (2004) Article DOI: 10.1021/jm0309912 BindingDB Entry DOI: 10.7270/Q26W9DS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413761![]() (CHEMBL390094) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cells | J Med Chem 45: 4391-4 (2002) Article DOI: 10.1021/jm025549i BindingDB Entry DOI: 10.7270/Q2FR00C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048691![]() (CHEMBL3315139) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413761![]() (CHEMBL390094) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413760![]() (CHEMBL426020) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50320463![]() (CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413760![]() (CHEMBL426020) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Salerno Curated by ChEMBL | Assay Description Binding affinity towards human Urotensin 2 receptor was determined | J Med Chem 47: 1652-61 (2004) Article DOI: 10.1021/jm0309912 BindingDB Entry DOI: 10.7270/Q26W9DS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413760![]() (CHEMBL426020) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cells | J Med Chem 45: 4391-4 (2002) Article DOI: 10.1021/jm025549i BindingDB Entry DOI: 10.7270/Q2FR00C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413764![]() (CHEMBL504097) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.282 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048696![]() (CHEMBL3315142) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.398 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048695![]() (CHEMBL3315141) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.724 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048701![]() (CHEMBL3315148) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.776 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413762![]() (CHEMBL509604) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.794 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50378580![]() (CHEMBL437430) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.794 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50378580![]() (CHEMBL437430) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.794 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Salerno Curated by ChEMBL | Assay Description Binding affinity towards human Urotensin 2 receptor was determined | J Med Chem 47: 1652-61 (2004) Article DOI: 10.1021/jm0309912 BindingDB Entry DOI: 10.7270/Q26W9DS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413784![]() (UROTENSIN-II) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | 0.794 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50378580![]() (CHEMBL437430) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.794 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cells | J Med Chem 45: 4391-4 (2002) Article DOI: 10.1021/jm025549i BindingDB Entry DOI: 10.7270/Q2FR00C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413766![]() (CHEMBL510618) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.891 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048700![]() (CHEMBL3315147) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048699![]() (CHEMBL3315146) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50473964![]() (CHEMBL2370836) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Salerno Curated by ChEMBL | Assay Description Binding affinity towards human Urotensin 2 receptor was determined | J Med Chem 47: 1652-61 (2004) Article DOI: 10.1021/jm0309912 BindingDB Entry DOI: 10.7270/Q26W9DS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50473964![]() (CHEMBL2370836) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cells | J Med Chem 45: 4391-4 (2002) Article DOI: 10.1021/jm025549i BindingDB Entry DOI: 10.7270/Q2FR00C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413763![]() (CHEMBL448403) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 1.66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048697![]() (CHEMBL3315144) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048705![]() (CHEMBL3315152) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048703![]() (CHEMBL3315150) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048692![]() (CHEMBL3315140) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048702![]() (CHEMBL3315149) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413777![]() (CHEMBL524855) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413769![]() (CHEMBL507406) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.89 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50411333![]() (URANTIDE) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50411333![]() (URANTIDE) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | Article PubMed | 5.01 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413770![]() (CHEMBL452403) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.46 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048690![]() (CHEMBL3315143) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413774![]() (CHEMBL509009) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413775![]() (CHEMBL501794) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413767![]() (CHEMBL504723) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413771![]() (CHEMBL509042) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048704![]() (CHEMBL3315151) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50474788![]() (CHEMBL2372643) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Salerno Curated by ChEMBL | Assay Description Binding affinity towards human Urotensin 2 receptor was determined | J Med Chem 47: 1652-61 (2004) Article DOI: 10.1021/jm0309912 BindingDB Entry DOI: 10.7270/Q26W9DS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048698![]() (CHEMBL3315145) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50473965![]() (CHEMBL2370837) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cells | J Med Chem 45: 4391-4 (2002) Article DOI: 10.1021/jm025549i BindingDB Entry DOI: 10.7270/Q2FR00C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413772![]() (CHEMBL508811) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413773![]() (CHEMBL500949) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 15.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50048706![]() (CHEMBL3315153) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples"Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting method | J Med Chem 57: 5965-74 (2014) Article DOI: 10.1021/jm500218x BindingDB Entry DOI: 10.7270/Q2MC91NB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413765![]() (CHEMBL501579) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413768![]() (CHEMBL505358) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Urotensin-2 receptor (Homo sapiens (Human)) | BDBM50413776![]() (CHEMBL505288) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 219 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples Federico II Curated by ChEMBL | Assay Description Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation counting | J Med Chem 52: 3927-40 (2009) Article DOI: 10.1021/jm900148c BindingDB Entry DOI: 10.7270/Q27W6DFT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA nucleotidylexotransferase (Homo sapiens (Human)) | BDBM50442248![]() (CHEMBL2441983) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sapienza" Universit£ di Roma Curated by ChEMBL | Assay Description Non-competitive inhibition of human TdT using 3'-OH as substrate | J Med Chem 56: 7431-41 (2013) Article DOI: 10.1021/jm4010187 BindingDB Entry DOI: 10.7270/Q2H70H8G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA nucleotidylexotransferase (Homo sapiens (Human)) | BDBM50442215![]() (CHEMBL2441974) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sapienza" Universit£ di Roma Curated by ChEMBL | Assay Description Competitive inhibition of human TdT using TTP as substrate | J Med Chem 56: 7431-41 (2013) Article DOI: 10.1021/jm4010187 BindingDB Entry DOI: 10.7270/Q2H70H8G | |||||||||||
More data for this Ligand-Target Pair |
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