Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153727![]() (CHEMBL3774695) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153737![]() (CHEMBL3774786) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153735![]() (CHEMBL3774970) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153725![]() (CHEMBL3775153) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents | Article PubMed | 240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153733![]() (CHEMBL3775128) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153736![]() (CHEMBL3775201) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153718![]() (CHEMBL450532) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50088574![]() (CHEMBL3577218) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 290 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 transfected in mouse NIH/3T3 MDR1-G185 cells assessed as reduction in daunomycin accumulation after 30 mins by flow cytometr... | J Nat Prod 78: 736-45 (2015) Article DOI: 10.1021/np500903a BindingDB Entry DOI: 10.7270/Q2VX0J7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153719![]() (CHEMBL499498) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 290 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153721![]() (CHEMBL3775788) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50154916![]() (CHEMBL3775786) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153723![]() (CHEMBL3775488) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 320 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353597![]() (CHEMBL1829396) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353602![]() (CHEMBL1829522) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353600![]() (CHEMBL1829520) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50154912![]() (CHEMBL3774875) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153724![]() (CHEMBL3774484) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 410 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153734![]() (CHEMBL3775696) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50088576![]() (CHEMBL3577215) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 transfected in mouse NIH/3T3 MDR1-G185 cells assessed as reduction in daunomycin accumulation after 30 mins by flow cytometr... | J Nat Prod 78: 736-45 (2015) Article DOI: 10.1021/np500903a BindingDB Entry DOI: 10.7270/Q2VX0J7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50275947![]() ((5S,14R,19S,28R)-10,23-dimethoxy-4,4,29,29-tetrame...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Orgánica Antonio González Curated by ChEMBL | Assay Description Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometry | J Med Chem 51: 7132-43 (2009) Article DOI: 10.1021/jm800403b BindingDB Entry DOI: 10.7270/Q2TB16R7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153738![]() (CHEMBL3775556) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50154913![]() (CHEMBL3775570) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353599![]() (CHEMBL1829518) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153726![]() (CHEMBL3774590) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50154911![]() (CHEMBL3775215) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153731![]() (CHEMBL3775149) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50275948![]() ((4R,13S,19R,28R)-8,23-dimethoxy-14,14,29,29-tetram...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 510 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Orgánica Antonio González Curated by ChEMBL | Assay Description Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometry | J Med Chem 51: 7132-43 (2009) Article DOI: 10.1021/jm800403b BindingDB Entry DOI: 10.7270/Q2TB16R7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353601![]() (CHEMBL1829521) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 510 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153732![]() (CHEMBL3775564) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 520 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153722![]() (CHEMBL3774613) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221858![]() ((1S,2R,4S,5R,6R,7S,9R,12R)-5-(acetyloxy)-12-[(fura...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 570 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353604![]() (CHEMBL1829527) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | 570 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221830![]() (CHEMBL394980 | nicotinic acid (1S,2R,4S,5R,6R,7S,9...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 580 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353598![]() (CHEMBL1829397) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 590 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153730![]() (CHEMBL3775566) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50088575![]() (CHEMBL3577217) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 610 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 transfected in mouse NIH/3T3 MDR1-G185 cells assessed as reduction in daunomycin accumulation after 30 mins by flow cytometr... | J Nat Prod 78: 736-45 (2015) Article DOI: 10.1021/np500903a BindingDB Entry DOI: 10.7270/Q2VX0J7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50088575![]() (CHEMBL3577217) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 610 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153739![]() (CHEMBL3775573) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 610 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50154915![]() (CHEMBL3775674) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221873![]() ((1S,2R,4S,5R,6R,7S,9R,12R)-5,12-bis(acetyloxy)-6-[...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50153885![]() (CHEMBL3775652) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica"Antonio Gonz£lez" Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH/3T3 cells assessed as inhibition of daunomycin efflux incubated for 30 mins by flow cytometry | J Med Chem 59: 1880-90 (2016) Article DOI: 10.1021/acs.jmedchem.5b01429 BindingDB Entry DOI: 10.7270/Q2CN75R5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50353603![]() (CHEMBL1829524) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 640 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 expressed in mouse NIH-3T3 cells assessed as daunomycin efflux after 30 mins by flow cytometry | Eur J Med Chem 46: 4915-23 (2011) Article DOI: 10.1016/j.ejmech.2011.07.048 BindingDB Entry DOI: 10.7270/Q2N29XB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221866![]() ((1S,2R,4S,5R,6R,7S,9R,12R)-5-(acetyloxy)-4-(benzoy...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221823![]() (CHEMBL234334 | nicotinic acid (1S,2R,4S,5R,6R,7S,9...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 710 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221872![]() ((1R,2R,3S,4S,5R,6R,7R,8S,9S)-3,4-bis(acetyloxy)-7,...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 730 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50275945![]() ((1R,2R,4R,7bR,9R,11aR)-2,5,5,9,12,12-Hexamethyl-1,...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 770 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Orgánica Antonio González Curated by ChEMBL | Assay Description Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometry | J Med Chem 51: 7132-43 (2009) Article DOI: 10.1021/jm800403b BindingDB Entry DOI: 10.7270/Q2TB16R7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50088577![]() (CHEMBL3577214) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 780 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez Curated by ChEMBL | Assay Description Inhibition of human MDR1 transfected in mouse NIH/3T3 MDR1-G185 cells assessed as reduction in daunomycin accumulation after 30 mins by flow cytometr... | J Nat Prod 78: 736-45 (2015) Article DOI: 10.1021/np500903a BindingDB Entry DOI: 10.7270/Q2VX0J7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221831![]() (CHEMBL394284 | furan-2-carboxylic acid (1S,2R,4S,5...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221825![]() ((1S,2R,4S,5R,6S,7R,8S,9R,12R)-4,12-bis(acetyloxy)-...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 910 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50221856![]() (CHEMBL412860 | furan-2-carboxylic acid (1S,2R,4S,5...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 960 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Instituto Universitario de Bio-OrgAnica Antonio GonzAlez Curated by ChEMBL | Assay Description Inhibition of human Pgp-mediated DNR transport in NIH3T3 cells by microplate assay | J Med Chem 50: 4808-17 (2007) Article DOI: 10.1021/jm070290v BindingDB Entry DOI: 10.7270/Q2K35TCP | |||||||||||
More data for this Ligand-Target Pair |
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