Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259245 (CHEMBL4064127 | US10266550, Compound 17a) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 970 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259244 (CHEMBL4076393 | US10266550, Compound 16) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259247 (CHEMBL4065223 | US10266550, Compound 11g) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259215 (CHEMBL4064887 | US10266550, Compound 11b) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259248 (CHEMBL4104625 | US10266550, Compound 17bbSelectivi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259242 (CHEMBL4072011 | US10266550, Compound 11e) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259214 (CHEMBL4061346 | US10266550, Compound 11a) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496611 (CHEMBL3134416) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496611 (CHEMBL3134416) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259221 (CHEMBL4097472 | US10266550, Compound 11d) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.56E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496611 (CHEMBL3134416) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496611 (CHEMBL3134416) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496604 (CHEMBL3134406) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259213 (CHEMBL4079855 | US10266550, Compound 7e) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496622 (CHEBI:34640 | CHEMBL1739417) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496617 (CHEMBL3134419) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.25E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496607 (CHEMBL3134407) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496617 (CHEMBL3134419) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496620 (CHEMBL3134413) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496619 (CHEMBL3134412) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496609 (CHEMBL3134418) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50061625 (4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496606 (CHEMBL3134409) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496612 (CHEMBL3134410) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496605 (CHEMBL3134411) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496621 (CHEMBL3134405) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496618 (CHEMBL3134408) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496614 (CHEMBL3134421) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259246 (CHEMBL4066307 | US10266550, Compound 10a) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50052414 (4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496609 (CHEMBL3134418) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496614 (CHEMBL3134421) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496613 (CHEMBL3134404) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50259212 (CHEMBL2002459 | US10266550, Compound 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawaii at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase-2alpha assessed as reduction in enzyme-mediated decatenation using kinetoplast DNA as substrate after 15 mins by et... | Eur J Med Chem 125: 515-527 (2017) Article DOI: 10.1016/j.ejmech.2016.09.053 BindingDB Entry DOI: 10.7270/Q2445PXH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496616 (CHEMBL3134415) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496615 (CHEMBL3134417) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496610 (CHEMBL3134420) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496616 (CHEMBL3134415) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496615 (CHEMBL3134417) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496608 (CHEBI:66955 | CHEMBL3134414) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 1 (Yersinia pestis) | BDBM50496613 (CHEMBL3134404) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of Yersinia pestis topoisomerase 1-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496610 (CHEMBL3134420) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA topoisomerase 2-alpha (Homo sapiens (Human)) | BDBM50496608 (CHEBI:66955 | CHEMBL3134414) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Hawai'i at Hilo Curated by ChEMBL | Assay Description Inhibition of human topoisomerase 2 alpha-mediated relaxation of supercoiled plasmid DNA by agarose gel electrophoresis | Medchemcomm 4: (2013) Article DOI: 10.1039/C3MD00238A BindingDB Entry DOI: 10.7270/Q23F4SM4 | |||||||||||
More data for this Ligand-Target Pair |