Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50241132 (3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 0.135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50241132 (3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 0.141 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50241132 (3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 0.178 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50241132 (3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 0.209 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM82423 (CAS_132947 | NSC_132947 | TRIPITRAMINE) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 0.302 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50241132 (3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 0.324 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50415153 (CHEMBL569307) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.692 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50415145 (CHEMBL571121) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50415144 (CHEMBL583051) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50530219 (CHEMBL4454983) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florence Curated by ChEMBL | Assay Description Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometry | J Med Chem 62: 1887-1901 (2019) Article DOI: 10.1021/acs.jmedchem.8b01372 BindingDB Entry DOI: 10.7270/Q2PR80F8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50530219 (CHEMBL4454983) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florence Curated by ChEMBL | Assay Description Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometry | J Med Chem 62: 1887-1901 (2019) Article DOI: 10.1021/acs.jmedchem.8b01372 BindingDB Entry DOI: 10.7270/Q2PR80F8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415153 (CHEMBL569307) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.51 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50415153 (CHEMBL569307) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415145 (CHEMBL571121) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50415152 (CHEMBL569760) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.09 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415153 (CHEMBL569307) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM39341 (11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 2.82 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M1 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50412182 (CHEMBL539120) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50412182 (CHEMBL539120) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50412182 (CHEMBL539120) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50412182 (CHEMBL539120) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50415145 (CHEMBL571121) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412313 (CHEMBL2021478) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM82423 (CAS_132947 | NSC_132947 | TRIPITRAMINE) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 3.55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M1 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412315 (CHEMBL2021476) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50415145 (CHEMBL571121) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412177 (CHEMBL493979) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412177 (CHEMBL493979) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50412182 (CHEMBL539120) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50412182 (CHEMBL539120) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50415153 (CHEMBL569307) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412312 (CHEMBL2021479) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415145 (CHEMBL571121) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.57 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50412314 (CHEMBL2021477) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50412313 (CHEMBL2021478) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M1 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50415158 (CHEMBL569712) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.61 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415144 (CHEMBL583051) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50415144 (CHEMBL583051) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.08 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415152 (CHEMBL569760) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415144 (CHEMBL583051) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.76 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415158 (CHEMBL569712) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.91 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50415154 (CHEMBL568870) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415154 (CHEMBL568870) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50412176 (CHEMBL493980) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50412176 (CHEMBL493980) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells | Bioorg Med Chem 16: 5490-500 (2008) Article DOI: 10.1016/j.bmc.2008.04.013 BindingDB Entry DOI: 10.7270/Q21N82BT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415152 (CHEMBL569760) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10.2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50530216 (CHEMBL4582201) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florence Curated by ChEMBL | Assay Description Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometry | J Med Chem 62: 1887-1901 (2019) Article DOI: 10.1021/acs.jmedchem.8b01372 BindingDB Entry DOI: 10.7270/Q2PR80F8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Rattus norvegicus (Rat)) | BDBM50530216 (CHEMBL4582201) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Florence Curated by ChEMBL | Assay Description Displacement of [3H]-methyllycaconitine from alpha7* nAChR in rat brain P2 membranes after 2.5 hrs by liquid scintillation spectrometry | J Med Chem 62: 1887-1901 (2019) Article DOI: 10.1021/acs.jmedchem.8b01372 BindingDB Entry DOI: 10.7270/Q2PR80F8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50415152 (CHEMBL569760) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universita di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation counting | J Med Chem 53: 201-7 (2010) Article DOI: 10.1021/jm901048j BindingDB Entry DOI: 10.7270/Q2D79CPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM82423 (CAS_132947 | NSC_132947 | TRIPITRAMINE) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 11.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Alma Mater Studiorum-University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M4 receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 7311-20 (2008) Article DOI: 10.1016/j.bmc.2008.06.025 BindingDB Entry DOI: 10.7270/Q24F1S07 | |||||||||||
More data for this Ligand-Target Pair |
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