Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nischarin (RAT) | BDBM50387827 (CHEMBL2058635) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50387827 (CHEMBL2058635) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.219 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]paraiodoclonidine from imidazoline I1 receptor in rat PC12 cells after 30 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM215802 (US9303019, 8) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.220 | -57.3 | n/a | n/a | n/a | n/a | n/a | 7.35 | 37 |
UNIVERSITE DE STRASBOURG US Patent | Assay Description Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ... | US Patent US9303019 (2016) BindingDB Entry DOI: 10.7270/Q2N878NR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070374 (CHEMBL3408293) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.220 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50179395 (CHEMBL14640) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | 0.891 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membrane | J Med Chem 45: 32-40 (2002) Article DOI: 10.1021/jm0110082 BindingDB Entry DOI: 10.7270/Q21N83VZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50179395 (CHEMBL14640) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | 0.891 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50387823 (CHEMBL2058631) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.930 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50387823 (CHEMBL2058631) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.933 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]paraiodoclonidine from imidazoline I1 receptor in rat PC12 cells after 30 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50091345 (CHEMBL2092861) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cells | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50138500 (2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50138500 (2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 42: 2737-40 (1999) Article DOI: 10.1021/jm991049m BindingDB Entry DOI: 10.7270/Q2KW5JR7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50138499 (2-Phenethyl-4,5-dihydro-1H-imidazole | CHEMBL14210) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM215805 (US9303019, 20) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.80 | -50.8 | n/a | n/a | n/a | n/a | n/a | 7.35 | 37 |
UNIVERSITE DE STRASBOURG US Patent | Assay Description Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ... | US Patent US9303019 (2016) BindingDB Entry DOI: 10.7270/Q2N878NR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070366 (CHEMBL3408289) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM215803 (US9303019, 9) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.80 | -50.8 | n/a | n/a | n/a | n/a | n/a | 7.35 | 37 |
UNIVERSITE DE STRASBOURG US Patent | Assay Description Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ... | US Patent US9303019 (2016) BindingDB Entry DOI: 10.7270/Q2N878NR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070375 (CHEMBL3408294) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070372 (CHEMBL3408291) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50016897 (2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821002 from human alpha2 adrenoceptor expressed in CHO cell membranes after 60 mins | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50091347 (CHEMBL71429) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cells | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070329 (CHEMBL268734) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50472306 (CHEMBL93845) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50472306 (CHEMBL93845) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 42: 2737-40 (1999) Article DOI: 10.1021/jm991049m BindingDB Entry DOI: 10.7270/Q2KW5JR7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070361 (CHEMBL3408298) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070330 (CHEMBL3408297) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM215800 (US9303019, 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 8.10 | -48.0 | n/a | n/a | n/a | n/a | n/a | 7.35 | 37 |
UNIVERSITE DE STRASBOURG US Patent | Assay Description Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ... | US Patent US9303019 (2016) BindingDB Entry DOI: 10.7270/Q2N878NR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50016897 (2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821001 from human alpha2A adrenoceptor expressed in CHO cells after 60 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50016897 (2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821001 from human alpha2C adrenoceptor expressed in CHO cells after 60 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50262235 (rilmenidine) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]paraiodoclonidine from imidazoline I1 receptor in rat PC12 cells after 30 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50179398 (CHEMBL94022) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranes | J Med Chem 42: 2737-40 (1999) Article DOI: 10.1021/jm991049m BindingDB Entry DOI: 10.7270/Q2KW5JR7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50179398 (CHEMBL94022) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cells | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50179398 (CHEMBL94022) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranes | J Med Chem 42: 2737-40 (1999) Article DOI: 10.1021/jm991049m BindingDB Entry DOI: 10.7270/Q2KW5JR7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50412250 (CHEMBL128168) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat cortex membrane | J Med Chem 45: 32-40 (2002) Article DOI: 10.1021/jm0110082 BindingDB Entry DOI: 10.7270/Q21N83VZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50262235 (rilmenidine) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821001 from human alpha2C adrenoceptor expressed in CHO cells after 60 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50016897 (2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50472305 (CHEMBL67706) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cells | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM215801 (US9303019, 5) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 19 | -45.8 | n/a | n/a | n/a | n/a | n/a | 7.35 | 37 |
UNIVERSITE DE STRASBOURG US Patent | Assay Description Binding assays were performed at 37° C. using [125I]LNP 911 as radioligand following the general procedure described but adapted to washed whole ... | US Patent US9303019 (2016) BindingDB Entry DOI: 10.7270/Q2N878NR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50138500 (2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranes | J Med Chem 42: 2737-40 (1999) Article DOI: 10.1021/jm991049m BindingDB Entry DOI: 10.7270/Q2KW5JR7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070373 (CHEMBL3408292) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50138500 (2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cells | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070364 (CHEMBL3408285) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50472305 (CHEMBL67706) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | J Med Chem 46: 2169-76 (2003) Article DOI: 10.1021/jm021113r BindingDB Entry DOI: 10.7270/Q2HH6NSW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50472306 (CHEMBL93845) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Predicted affinity for imidazoline receptor I2 by three field CoMFA model | J Med Chem 42: 2737-40 (1999) Article DOI: 10.1021/jm991049m BindingDB Entry DOI: 10.7270/Q2KW5JR7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070363 (CHEMBL3408284) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50016897 (2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821001 from human alpha2B adrenoceptor expressed in CHO cells after 60 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473618 (CHEMBL337945) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat cortex membrane | J Med Chem 45: 32-40 (2002) Article DOI: 10.1021/jm0110082 BindingDB Entry DOI: 10.7270/Q21N83VZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50417354 (CHEMBL396013) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat cortex membrane | J Med Chem 45: 32-40 (2002) Article DOI: 10.1021/jm0110082 BindingDB Entry DOI: 10.7270/Q21N83VZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A/B (Homo sapiens (Human)) | BDBM50473129 (Phenamazoline) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membrane | J Med Chem 45: 32-40 (2002) Article DOI: 10.1021/jm0110082 BindingDB Entry DOI: 10.7270/Q21N83VZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50262235 (rilmenidine) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821001 from human alpha2A adrenoceptor expressed in CHO cells after 60 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (RAT) | BDBM50070368 (CHEMBL3408290) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 42 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma counting | J Med Chem 58: 878-87 (2015) Article DOI: 10.1021/jm501456p BindingDB Entry DOI: 10.7270/Q2R21333 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50262235 (rilmenidine) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ de Strasbourg Curated by ChEMBL | Assay Description Displacement of [3H]RX821001 from human alpha2B adrenoceptor expressed in CHO cells after 60 mins by gamma counter | Bioorg Med Chem 20: 4710-5 (2012) Article DOI: 10.1016/j.bmc.2012.06.008 BindingDB Entry DOI: 10.7270/Q26Q1Z9Q | |||||||||||
More data for this Ligand-Target Pair |
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