Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aromatase [1-48] (Homo sapiens (Human)) | BDBM13061 (4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Biomolécules et Cibles Cellulaires Tumorales | Assay Description The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion... | Bioorg Chem 32: 494-503 (2004) Article DOI: 10.1016/j.bioorg.2004.06.008 BindingDB Entry DOI: 10.7270/Q21R6P2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50118965 (4-Imidazol-1-yl-2-phenyl-chroman-7-ol | CHEMBL9591...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Biomolécules et Cibles Cellulaires Tumorales Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomes | Bioorg Med Chem Lett 14: 5215-8 (2004) Article DOI: 10.1016/j.bmcl.2004.07.090 BindingDB Entry DOI: 10.7270/Q26Q1WQ8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase [1-48] (Homo sapiens (Human)) | BDBM85252 (2,4-Trans-4'-hydroxy-4-imidazolyl-7-methoxyfla...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Biomolécules et Cibles Cellulaires Tumorales | Assay Description The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion... | Bioorg Chem 32: 494-503 (2004) Article DOI: 10.1016/j.bioorg.2004.06.008 BindingDB Entry DOI: 10.7270/Q21R6P2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50118965 (4-Imidazol-1-yl-2-phenyl-chroman-7-ol | CHEMBL9591...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description Inhibition of aromatase activity in human placental microsomes | Bioorg Med Chem Lett 12: 2859-61 (2002) BindingDB Entry DOI: 10.7270/Q2PK0FHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase [1-48] (Homo sapiens (Human)) | BDBM85253 (2,4-Trans-4',7-dihydroxy-4-imidazolyl-7-methox...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 77 | n/a | n/a | n/a | n/a | n/a | n/a |
Biomolécules et Cibles Cellulaires Tumorales | Assay Description The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion... | Bioorg Chem 32: 494-503 (2004) Article DOI: 10.1016/j.bioorg.2004.06.008 BindingDB Entry DOI: 10.7270/Q21R6P2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50118966 (1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Biomolécules et Cibles Cellulaires Tumorales Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomes | Bioorg Med Chem Lett 14: 5215-8 (2004) Article DOI: 10.1016/j.bmcl.2004.07.090 BindingDB Entry DOI: 10.7270/Q26Q1WQ8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50118966 (1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 91 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description Inhibition of aromatase activity in human placental microsomes | Bioorg Med Chem Lett 12: 2859-61 (2002) BindingDB Entry DOI: 10.7270/Q2PK0FHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase [1-48] (Homo sapiens (Human)) | BDBM85249 (2,4-Trans-3'-hydroxy-4-imidazolyl-7-methoxyfla...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Biomolécules et Cibles Cellulaires Tumorales | Assay Description The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion... | Bioorg Chem 32: 494-503 (2004) Article DOI: 10.1016/j.bioorg.2004.06.008 BindingDB Entry DOI: 10.7270/Q21R6P2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase [1-48] (Homo sapiens (Human)) | BDBM85251 (2,4-Trans-4'-cyano-4-imidazolyl-7-methoxyflava...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 133 | n/a | n/a | n/a | n/a | n/a | n/a |
Biomolécules et Cibles Cellulaires Tumorales | Assay Description The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion... | Bioorg Chem 32: 494-503 (2004) Article DOI: 10.1016/j.bioorg.2004.06.008 BindingDB Entry DOI: 10.7270/Q21R6P2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase [1-48] (Homo sapiens (Human)) | BDBM85250 (2,4-Trans-4'-chloro-4-imidazolyl-7-methoxyflav...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Biomolécules et Cibles Cellulaires Tumorales | Assay Description The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion... | Bioorg Chem 32: 494-503 (2004) Article DOI: 10.1016/j.bioorg.2004.06.008 BindingDB Entry DOI: 10.7270/Q21R6P2Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50153525 (2-Phenyl-4-[1,2,4]triazol-1-yl-chroman-7-ol | CHEM...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Biomolécules et Cibles Cellulaires Tumorales Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomes | Bioorg Med Chem Lett 14: 5215-8 (2004) Article DOI: 10.1016/j.bmcl.2004.07.090 BindingDB Entry DOI: 10.7270/Q26Q1WQ8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50374254 (CHEMBL439241) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50111269 (7-Methoxy-2-phenyl-3-pyridin-4-ylmethylene-chroman...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50345188 (2-(4-hydroxyphenyl)-2,3-dihydrobenzo[h]chromen-4-o...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50111268 (2-Phenyl-3-pyridin-4-ylmethylene-chroman-4-one | C...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50374255 (CHEMBL258257) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50153523 (1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-[1,2,4]tria...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Biomolécules et Cibles Cellulaires Tumorales Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomes | Bioorg Med Chem Lett 14: 5215-8 (2004) Article DOI: 10.1016/j.bmcl.2004.07.090 BindingDB Entry DOI: 10.7270/Q26Q1WQ8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50345187 (4-(4-oxo-3,4-dihydro-2H-benzo[h]chromen-2-yl)benzo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50111270 (7-Methoxy-2-phenyl-3-pyridin-4-ylmethylene-chroman...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50014323 (2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50241408 ((2S)-liquiritigenin | 7-HYDROXY-2-(4-HYDROXY-PHENY...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50111271 (2-Phenyl-3-pyridin-4-ylmethylene-chroman-4-one | C...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50374256 (CHEMBL255110) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50374258 (CHEMBL256407) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50374257 (CHEMBL402970) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50104887 (2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50104887 (2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description Inhibition of aromatase activity in human placental microsomes | Bioorg Med Chem Lett 12: 2859-61 (2002) BindingDB Entry DOI: 10.7270/Q2PK0FHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50345186 (2-phenyl-2,3-dihydrobenzo[h]chromen-4-one | 2-phen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM9460 (3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description Inhibition of aromatase activity in human placental microsomes | Bioorg Med Chem Lett 12: 2859-61 (2002) BindingDB Entry DOI: 10.7270/Q2PK0FHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM9460 (3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50106920 ((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description Inhibition of aromatase activity in human placental microsomes | Bioorg Med Chem Lett 12: 2859-61 (2002) BindingDB Entry DOI: 10.7270/Q2PK0FHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50106920 ((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50106920 ((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50051358 (2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50051358 (2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1 | Bioorg Med Chem Lett 12: 1059-61 (2002) BindingDB Entry DOI: 10.7270/Q2125S01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50153524 (4-(7-Methoxy-2-phenyl-chroman-4-yl)-4H-[1,2,4]tria...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.16E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Biomolécules et Cibles Cellulaires Tumorales Curated by ChEMBL | Assay Description In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomes | Bioorg Med Chem Lett 14: 5215-8 (2004) Article DOI: 10.1016/j.bmcl.2004.07.090 BindingDB Entry DOI: 10.7270/Q26Q1WQ8 | |||||||||||
More data for this Ligand-Target Pair |