Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50089314 (CHEMBL405182 | H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin. | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50089316 (CHEMBL410068 | H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity of the compound towards human cloned B1 receptor was determined using [3H]-[des-Arg10-Leu9]-kallidin as radioligand | J Med Chem 43: 2387-94 (2000) BindingDB Entry DOI: 10.7270/Q2N87913 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50089307 (CHEMBL410579 | H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin. | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50403371 (Firazyr | HOE-140 | ICATIBANT) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | PubMed | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement. | J Med Chem 42: 4193-201 (1999) BindingDB Entry DOI: 10.7270/Q2222VFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50403371 (Firazyr | HOE-140 | ICATIBANT) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | PubMed | 0.0640 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand | J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement. | J Med Chem 42: 4193-201 (1999) BindingDB Entry DOI: 10.7270/Q2222VFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50081659 ((3-(Ser-Thi-Gly-Hyp-Pro-Arg-Lys-H)-4-oxo-3,4-dihyd...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement. | J Med Chem 42: 4193-201 (1999) BindingDB Entry DOI: 10.7270/Q2222VFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50403371 (Firazyr | HOE-140 | ICATIBANT) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | PubMed | 0.0770 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligand | J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50089308 (CHEMBL412349 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykinin | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykinin | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420581 (CHEMBL2087422) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50089313 (CHEMBL412824 | H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.220 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin. | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50326708 (CHEMBL1254771 | N-(4-(4,5-dihydro-1H-imidazol-2-yl...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50089313 (CHEMBL412824 | H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykinin | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420570 (CHEMBL2087434) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity against rat Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand | J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand | J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420569 (CHEMBL2087433) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50408748 (CHEMBL2112698) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand | J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50081660 ((JMV 1116) H-D-Arg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-Ar...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement. | J Med Chem 42: 4193-201 (1999) BindingDB Entry DOI: 10.7270/Q2222VFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420579 (CHEMBL2087423) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50089310 (2-({1-[2-(2-{2-[(1-{1-[2-(2,6-Diamino-hexanoylamin...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin. | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420589 (CHEMBL2087031) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Binding affinity to B1 receptor | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor A (RAT) | BDBM50082568 (2-({3-[4-(2-Azido-benzenesulfonylaminocarbonyl)-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier S.A. Curated by ChEMBL | Assay Description The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes. | J Med Chem 42: 4572-83 (1999) BindingDB Entry DOI: 10.7270/Q2XW4J1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420580 (CHEMBL2087421) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420603 (CHEMBL2087035) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Type-1 angiotensin II receptor A (RAT) | BDBM50082567 (2-({2-Butyl-3-[4-(2-chloro-benzenesulfonylaminocar...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier S.A. Curated by ChEMBL | Assay Description The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes. | J Med Chem 42: 4572-83 (1999) BindingDB Entry DOI: 10.7270/Q2XW4J1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50081663 ((3-(Ser-Thi-Gly-Hyp-Pro-Arg-D-Arg-H)-4-oxo-3,4-dih...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement. | J Med Chem 42: 4193-201 (1999) BindingDB Entry DOI: 10.7270/Q2222VFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420595 (CHEMBL2087409) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420597 (CHEMBL2087411) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420582 (CHEMBL2087420) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420573 (CHEMBL2087429) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420571 (CHEMBL2087432) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420601 (CHEMBL2087412) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420598 (CHEMBL2087413) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50089312 (CHEMBL408846 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykinin | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420577 (CHEMBL2087424) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420568 (CHEMBL2087435) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420596 (CHEMBL2087410) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420583 (CHEMBL2087418) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50089309 (CHEMBL216618 | H-DArg-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin. | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420574 (CHEMBL2087427) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (RAT) | BDBM50408748 (CHEMBL2112698) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligand | J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50081662 ((3-(Ser-Thi-Gly-Hyp-Pro-Arg-D-Arg-H),-8-methyl-4-o...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£s Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement. | J Med Chem 42: 4193-201 (1999) BindingDB Entry DOI: 10.7270/Q2222VFV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420600 (CHEMBL2087415) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50089316 (CHEMBL410068 | H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Binding affinity of the compound towards human cloned B2 receptor was determined using [3H]-BK as radioligand | J Med Chem 43: 2387-94 (2000) BindingDB Entry DOI: 10.7270/Q2N87913 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50089314 (CHEMBL405182 | H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykinin | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420572 (CHEMBL2087431) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | >10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universités Montpellier I et II Curated by ChEMBL | Assay Description Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin. | J Med Chem 43: 2382-6 (2000) BindingDB Entry DOI: 10.7270/Q2S181QZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Homo sapiens (Human)) | BDBM50420575 (CHEMBL2087428) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratoires Fournier Curated by ChEMBL | Assay Description Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counter | J Med Chem 55: 2574-84 (2012) Article DOI: 10.1021/jm2016057 BindingDB Entry DOI: 10.7270/Q20C4X1J | |||||||||||
More data for this Ligand-Target Pair |
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