Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468736 (US10807959, Example 5) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473225 (US10844044, Example 283) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468925 (US10807959, Example B64) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476247 (CHEMBL224081) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.A. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cells | J Med Chem 47: 6935-47 (2004) Article DOI: 10.1021/jm040832y BindingDB Entry DOI: 10.7270/Q2T43WVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388901 (CHEMBL2063237) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced [35S]GTPgammaS binding incubated for 1... | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468927 (US10807959, Example B74) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468928 (US10807959, Example B81) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0330 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468938 (US10807959, Example B109) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388885 (CHEMBL2063238) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced [35S]GTPgammaS binding incubated for 1... | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM50520121 (CHEMBL4441671 | US10844044, Example 1) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | 0.0440 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Frederick National Laboratory for Cancer Research Curated by ChEMBL | Assay Description Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer... | J Med Chem 63: 656-675 (2020) Article DOI: 10.1021/acs.jmedchem.9b01608 BindingDB Entry DOI: 10.7270/Q2HD801W | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50404016 (CHEMBL2112922) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.A. Laboratori di Firenze Curated by ChEMBL | Assay Description In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB) | Bioorg Med Chem Lett 12: 693-6 (2002) BindingDB Entry DOI: 10.7270/Q22N53FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473480 (US10844044, Example 72) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388902 (CHEMBL2063239) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced [35S]GTPgammaS binding incubated for 1... | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50404016 (CHEMBL2112922) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0501 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.A. Laboratori di Firenze Curated by ChEMBL | Assay Description In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB) | Bioorg Med Chem Lett 12: 693-6 (2002) BindingDB Entry DOI: 10.7270/Q22N53FR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476235 (CHEMBL436981) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0501 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.A. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cells | J Med Chem 47: 6935-47 (2004) Article DOI: 10.1021/jm040832y BindingDB Entry DOI: 10.7270/Q2T43WVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476788 (CHEMBL243711) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0525 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.a. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human recombinant NK2 receptor | J Med Chem 50: 4793-807 (2007) Article DOI: 10.1021/jm070289w BindingDB Entry DOI: 10.7270/Q2CR5X4G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476771 (CHEMBL244362) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0575 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.a. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human recombinant NK2 receptor | J Med Chem 50: 4793-807 (2007) Article DOI: 10.1021/jm070289w BindingDB Entry DOI: 10.7270/Q2CR5X4G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473383 (US10844044, Example 230) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473215 (US10844044, Example 98) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473393 (US10844044, Example 232) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476748 (CHEMBL395972) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0603 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.a. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human recombinant NK2 receptor | J Med Chem 50: 4793-807 (2007) Article DOI: 10.1021/jm070289w BindingDB Entry DOI: 10.7270/Q2CR5X4G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476221 (CHEMBL387506) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.A. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cells | J Med Chem 47: 6935-47 (2004) Article DOI: 10.1021/jm040832y BindingDB Entry DOI: 10.7270/Q2T43WVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476233 (CHEMBL439281) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.A. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cells | J Med Chem 47: 6935-47 (2004) Article DOI: 10.1021/jm040832y BindingDB Entry DOI: 10.7270/Q2T43WVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Rattus norvegicus (rat)) | BDBM50130172 (1-(3-Benzo[b]thiophen-2-yl-8-aza-bicyclo[3.2.1]oct...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description In vitro affinity of the compound at the 5-HT reuptake site using [3H]-paroxetine as radioligand in rat frontal cortex membranes | Bioorg Med Chem Lett 13: 2393-7 (2003) BindingDB Entry DOI: 10.7270/Q2Z31Z1R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388887 (CHEMBL2063240) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced [35S]GTPgammaS binding incubated for 1... | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476750 (Ibodutant | MEN-15596) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | 0.0759 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.a. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human recombinant NK2 receptor | J Med Chem 50: 4793-807 (2007) Article DOI: 10.1021/jm070289w BindingDB Entry DOI: 10.7270/Q2CR5X4G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388893 (CHEMBL2063246) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced [35S]GTPgammaS binding incubated for 1... | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388896 (CHEMBL2063249) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP-55940-induced [35S]GTPgammaS binding incubated for 1... | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468936 (US10807959, Example B99) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0870 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468939 (US10807959, Example B111) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0870 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468945 (US10807959, Example B129) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0890 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50388887 (CHEMBL2063240) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]SR141716A form human CB1 receptor expressed in HEK293 cells after 60 mins by beta counting | ACS Med Chem Lett 3: 397-401 (2012) Article DOI: 10.1021/ml3000325 BindingDB Entry DOI: 10.7270/Q22N53BD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM468937 (US10807959, Example B107) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.0970 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr... | US Patent US10807959 (2020) BindingDB Entry DOI: 10.7270/Q26Q219X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (Homo sapiens (Human)) | BDBM50476764 (CHEMBL395974) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.0977 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche S.p.a. Curated by ChEMBL | Assay Description Displacement of [125I]neurokinin A from human recombinant NK2 receptor | J Med Chem 50: 4793-807 (2007) Article DOI: 10.1021/jm070289w BindingDB Entry DOI: 10.7270/Q2CR5X4G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473503 (US10844044, Example 352) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473507 (US10844044, Example 353) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473511 (US10844044, Example 354) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473517 (US10844044, Example 172) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473525 (US10844044, Example 174) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473532 (US10844044, Example 85) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473534 (US10844044, Example 268) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473538 (US10844044, Example 269) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473431 (US10844044, Example 334) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473432 (US10844044, Example 60) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473434 (US10844044, Example 242) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473435 (US10844044, Example 335) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473438 (US10844044, Example 243) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473439 (US10844044, Example 336) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473442 (US10844044, Example 244) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
WD repeat-containing protein 5 (Homo sapiens (Human)) | BDBM473443 (US10844044, Example 337) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <0.100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description A Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) assay that measures the displacement of the 10mer-Thr-FAM probe in response to compo... | US Patent US10844044 (2020) BindingDB Entry DOI: 10.7270/Q21R6TKB | |||||||||||
More data for this Ligand-Target Pair |
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