Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518898 (US11116757, No. A193) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <2.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM519032 (US11116757, No. B19) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM519034 (US11116757, No. B21) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50079170 (1-(1-Benzyl-piperidin-4-yl)-3-phenyl-urea | CHEMBL...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | <4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518647 (US11116757, No. A1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518656 (US11116757, No. A2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518671 (US11116757, No. A3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245227 (CHEMBL4077431 | US11116757, No. A4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245225 (CHEMBL4099097 | US11116757, No. A15) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245225 (CHEMBL4099097 | US11116757, No. A15) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245131 (CHEMBL4094517 | US11116757, No. A5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 55.9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245148 (CHEMBL4077759 | US11116757, No. A6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245237 (CHEMBL4074213 | US11116757, No. A7) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 76.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245153 (CHEMBL4078685 | US11116757, No. A8) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 76.7 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518705 (US11116757, No. A9) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 78.8 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245154 (CHEMBL4067795 | US11116757, No. A10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 78.9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245140 (CHEMBL4103209 | US11116757, No. A11) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 81.8 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518708 (US11116757, No. A12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 82.7 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245130 (CHEMBL4086099 | US11116757, No. A13) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518710 (US11116757, No. A14) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 85.3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245225 (CHEMBL4099097 | US11116757, No. A15) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 88.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518714 (US11116757, No. A16) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 90.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518715 (US11116757, No. A17) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 95.1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460825 (CHEMBL4102019 | US11116757, No. A21) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460825 (CHEMBL4102019 | US11116757, No. A21) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518716 (US11116757, No. A18) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 111 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518720 (US11116757, No. A20) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 116 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518718 (US11116757, No. A19) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 116 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460825 (CHEMBL4102019 | US11116757, No. A21) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 119 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460827 (CHEMBL4077751 | US11116757, No. A43) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518722 (US11116757, No. A22) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 131 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460853 (CHEMBL4229003 | US11116757, No. A37) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518725 (US11116757, No. A23) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518822 (US11116757, No. A118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 143 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518726 (US11116757, No. A24) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 154 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518727 (US11116757, No. A25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 155 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245223 (CHEMBL4085483 | US11116757, No. A26) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 163 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518729 (US11116757, No. A27) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 165 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245238 (CHEMBL4103413 | US11116757, No. A28) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 166 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50525343 (CHEMBL4440896 | US11116757, No. A29) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 172 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460829 (CHEMBL4225246 | US11116757, No. A30) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 178 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460829 (CHEMBL4225246 | US11116757, No. A30) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518733 (US11116757, No. A31) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 184 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518734 (US11116757, No. A32) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460836 (CHEMBL4072130 | US11116757, No. A34) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245226 (CHEMBL4093853 | US11116757, No. A33) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460836 (CHEMBL4072130 | US11116757, No. A34) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 201 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245117 (CHEMBL4077301 | US11116757, No. A35) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 202 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM518738 (US11116757, No. A36) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 206 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50460853 (CHEMBL4229003 | US11116757, No. A37) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 207 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 690 total ) | Next | Last >> |