BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Chymotrypsin-like protease CTRL-1' and Ligand = 'BDBM50288610'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Chymotrypsin-like protease CTRL-1 (Homo sapiens (Human))	BDBM50288610 (Alpha-ketocarbonyl derivative \| CHEMBL98937) Show SMILES Show InChI	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was tested for thromboxane TXA2 synthase inhibitory activity using human platelet				Bioorg Med Chem Lett 6: 287-290 (1996) Article DOI: 10.1016/0960-894X(96)00014-5 BindingDB Entry DOI: 10.7270/Q2JQ1112
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Chymotrypsin-like protease CTRL-1 (Homo sapiens (Human))	BDBM50288610 (Alpha-ketocarbonyl derivative \| CHEMBL98937) Show SMILES Show InChI	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brain				Bioorg Med Chem Lett 6: 287-290 (1996) Article DOI: 10.1016/0960-894X(96)00014-5 BindingDB Entry DOI: 10.7270/Q2JQ1112
TBA Curated by ChEMBL					More data for this Ligand-Target Pair