Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016504 ((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brain | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of 0.1 nM [3H]-pCCK-8 from guinea pig pancreatic membranes | J Med Chem 32: 1184-90 (1989) BindingDB Entry DOI: 10.7270/Q2ZG6R7N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to CCK-8 receptor of guinea pig brain | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor of Guinea pig pancreatic membranes | J Med Chem 40: 647-58 (1997) Article DOI: 10.1021/jm9603072 BindingDB Entry DOI: 10.7270/Q2PG1SDX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016504 ((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranes | Bioorg Med Chem Lett 14: 369-72 (2003) BindingDB Entry DOI: 10.7270/Q2RJ4K1Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranes | Bioorg Med Chem Lett 14: 369-72 (2003) BindingDB Entry DOI: 10.7270/Q2RJ4K1Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article | 0.640 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pig | Bioorg Med Chem Lett 3: 847-850 (1993) Article DOI: 10.1016/S0960-894X(00)80678-2 BindingDB Entry DOI: 10.7270/Q2P26Z28 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.640 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brain | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Compound was tested for binding affinity against CCK1 (cholecystokinin) receptor on guinea pig pancreatic membranes | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092398 ((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092405 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | >0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM21147 ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of [3H]-pCCK-8 from cholecystokinin-A receptor in guinea pig pancreatic membrane | J Med Chem 36: 166-72 (1993) BindingDB Entry DOI: 10.7270/Q26M37FJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092405 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranes | Bioorg Med Chem Lett 14: 369-72 (2003) BindingDB Entry DOI: 10.7270/Q2RJ4K1Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016504 ((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.930 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membrane | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016425 ((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.930 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of 0.1 nM [3H]-pCCK-8 from guinea pig pancreatic membranes | J Med Chem 32: 1184-90 (1989) BindingDB Entry DOI: 10.7270/Q2ZG6R7N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092388 (3-(2-{[2-(3-tert-Butoxycarbonylamino-propionylamin...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016506 (CHEMBL262687 | Sodium; (4-{2-(2-acetylamino-3-carb...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membrane | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092391 (3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.05 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092396 (3-(2-{[2-Amino-3-(1H-indol-3-yl)-propionyl]-methyl...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092398 ((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranes | Bioorg Med Chem Lett 14: 369-72 (2003) BindingDB Entry DOI: 10.7270/Q2RJ4K1Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50138278 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranes | Bioorg Med Chem Lett 14: 369-72 (2003) BindingDB Entry DOI: 10.7270/Q2RJ4K1Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016503 (Boc-Asp-D-Tyr(SO3Na)-Nle-Gly-Trp-Nle-Asp-Phe-NH2 |...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brain | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092384 (CHEMBL100538 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.02 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016506 (CHEMBL262687 | Sodium; (4-{2-(2-acetylamino-3-carb...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to CCK-8 receptor of guinea pig pancreatic membrane | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092402 (CHEMBL122872 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.35 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50046112 (3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-({[...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of [3H]-pCCK-8 from cholecystokinin-A receptor in guinea pig pancreatic membrane | J Med Chem 36: 166-72 (1993) BindingDB Entry DOI: 10.7270/Q26M37FJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092400 (3-(2-{[2-(2-Amino-propionylamino)-3-(1H-indol-3-yl...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092394 ((S)-3-((S)-2-{[(S)-2-(2-Amino-acetylamino)-3-(S)-1...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016505 (CHEMBL217767 | Sodium; (4-{2-(2-acetylamino-3-carb...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brain | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016505 (CHEMBL217767 | Sodium; (4-{2-(2-acetylamino-3-carb...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membrane | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092390 (3-(2-{[2-(2-Amino-propionylamino)-3-(1H-indol-3-yl...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016503 (Boc-Asp-D-Tyr(SO3Na)-Nle-Gly-Trp-Nle-Asp-Phe-NH2 |...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membrane | J Med Chem 32: 445-9 (1989) BindingDB Entry DOI: 10.7270/Q2S181GT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50281664 (CHEMBL262894 | p-Tyr(SO3Na)-gNle-mGly-Trp-(N-Me)Nl...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article | 62 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pig | Bioorg Med Chem Lett 3: 847-850 (1993) Article DOI: 10.1016/S0960-894X(00)80678-2 BindingDB Entry DOI: 10.7270/Q2P26Z28 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50477904 (CHEMBL401098) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 63 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cells | J Med Chem 51: 565-73 (2008) Article DOI: 10.1021/jm070880t BindingDB Entry DOI: 10.7270/Q2TF014R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50045802 (CHEMBL99252 | {[2-(Adamantan-2-yloxycarbonylamino)...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranes | J Med Chem 36: 2868-77 (1993) BindingDB Entry DOI: 10.7270/Q2MG7NK5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50016504 ((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pig | Bioorg Med Chem Lett 3: 847-850 (1993) Article DOI: 10.1016/S0960-894X(00)80678-2 BindingDB Entry DOI: 10.7270/Q2P26Z28 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50092393 (3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 96 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50228603 (CHEMBL3350278) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranes | J Med Chem 33: 3199-204 (1991) BindingDB Entry DOI: 10.7270/Q2XP73WF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50228604 (CHEMBL3350720) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranes | J Med Chem 33: 3199-204 (1991) BindingDB Entry DOI: 10.7270/Q2XP73WF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50056455 (CHEMBL348344 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 271 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor of Guinea pig pancreatic membranes | J Med Chem 40: 647-58 (1997) Article DOI: 10.1021/jm9603072 BindingDB Entry DOI: 10.7270/Q2PG1SDX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50470630 (CHEMBL436187) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 302 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Competition with 20 pM [125I]BH-CCK-8S at Cholecystokinin type A receptor binding sites on guinea pig pancreatic cells | J Med Chem 38: 4294-302 (1995) Article DOI: 10.1021/jm00021a019 BindingDB Entry DOI: 10.7270/Q2930WWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50470639 (CHEMBL433656) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 302 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Competition with 20 pM [125I]BH-CCK-8S at Cholecystokinin type A receptor binding sites on guinea pig pancreatic cells | J Med Chem 38: 4294-302 (1995) Article DOI: 10.1021/jm00021a019 BindingDB Entry DOI: 10.7270/Q2930WWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50228605 (CHEMBL3350665) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranes | J Med Chem 33: 3199-204 (1991) BindingDB Entry DOI: 10.7270/Q2XP73WF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50477908 (CHEMBL398312) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 316 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cells | J Med Chem 51: 565-73 (2008) Article DOI: 10.1021/jm070880t BindingDB Entry DOI: 10.7270/Q2TF014R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM81962 (S-L-365,260) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 316 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cells | J Med Chem 51: 565-73 (2008) Article DOI: 10.1021/jm070880t BindingDB Entry DOI: 10.7270/Q2TF014R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50228605 (CHEMBL3350665) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranes | J Med Chem 33: 3199-204 (1991) BindingDB Entry DOI: 10.7270/Q2XP73WF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50228602 (CHEMBL3350331) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranes | J Med Chem 33: 3199-204 (1991) BindingDB Entry DOI: 10.7270/Q2XP73WF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50469591 (CHEMBL288641) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article | 355 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description In vitro affinity against Cholecystokinin type A receptor in guinea pig pancreatic cell | Citation and Details Article DOI: 10.1016/S0960-894X(00)80008-6 BindingDB Entry DOI: 10.7270/Q2BC4270 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50056102 ((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 398 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cells | J Med Chem 51: 565-73 (2008) Article DOI: 10.1021/jm070880t BindingDB Entry DOI: 10.7270/Q2TF014R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50470640 (CHEMBL443028) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 447 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
James Black Foundation Curated by ChEMBL | Assay Description Competition with 20 pM [125I]BH-CCK-8S at Cholecystokinin type A receptor binding sites on guinea pig pancreatic cells | J Med Chem 38: 4294-302 (1995) Article DOI: 10.1021/jm00021a019 BindingDB Entry DOI: 10.7270/Q2930WWV | |||||||||||
More data for this Ligand-Target Pair |
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