Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50156455 ((R)-N-(4-(4,5-dihydro-1H-imidazol-2-yl)phenethyl)-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson& Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of rabbit bradykinin B1 receptor | J Med Chem 53: 5383-99 (2010) Article DOI: 10.1021/jm1000776 BindingDB Entry DOI: 10.7270/Q289162Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355062 (CHEMBL1834752) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355063 (CHEMBL1834619) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355057 (CHEMBL1834751) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50157515 (4'-{(R)-1-[4-chloro-3-(2-cyano-acetylamino)-pyridi...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Activity at rabbit bradykinin B1 receptor assessed by FLIPR assay | J Med Chem 47: 6439-42 (2004) Article DOI: 10.1021/jm049394l BindingDB Entry DOI: 10.7270/Q22B8XHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50157511 (CHEMBL387638 | N-(4-chloro-2-{(R)-1-[3'-fluoro-2'-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Activity at rabbit bradykinin B1 receptor assessed by FLIPR assay | J Med Chem 47: 6439-42 (2004) Article DOI: 10.1021/jm049394l BindingDB Entry DOI: 10.7270/Q22B8XHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50344100 (2-((2R)-1-((4-methylphenyl)sulfonyl)-3-oxo-2-piper...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50157513 (3-chloro-4'-{(R)-1-[4-chloro-3-(2-cyano-acetylamin...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Activity at rabbit bradykinin B1 receptor assessed by FLIPR assay | J Med Chem 47: 6439-42 (2004) Article DOI: 10.1021/jm049394l BindingDB Entry DOI: 10.7270/Q22B8XHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50209744 ((R)-3-(4-fluorophenyl)-N-((R)-7-(piperidin-1-ylmet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 10.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor | J Med Chem 50: 2200-12 (2007) Article DOI: 10.1021/jm070055c BindingDB Entry DOI: 10.7270/Q2MS3SG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244617 ((2R,3S)-2,3-dihydroxy-N-((R)-6-(piperidin-1-ylmeth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244617 ((2R,3S)-2,3-dihydroxy-N-((R)-6-(piperidin-1-ylmeth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50157509 (CHEMBL222038 | N-(4-chloro-2-{(R)-1-[3'-fluoro-2'-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Activity at rabbit bradykinin B1 receptor assessed by FLIPR assay | J Med Chem 47: 6439-42 (2004) Article DOI: 10.1021/jm049394l BindingDB Entry DOI: 10.7270/Q22B8XHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50203200 ((R)-3-(naphthalene-7-sulfonamido)-3-phenyl-N-((R)-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonistic activity at rabbit bradykinin B1 receptor expressed in CHO-D cells assessed as effect on DAK-mediated calcium mobilization | J Med Chem 50: 607-10 (2007) Article DOI: 10.1021/jm061224g BindingDB Entry DOI: 10.7270/Q2KP81T0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355058 (CHEMBL1834750) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 17.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244566 ((2R,3S)-2,3-dihydroxy-4-(naphthalen-2-ylsulfonyl)-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244438 ((2R,3S)-4-(3,4-dichlorophenylsulfonyl)-2,3-dihydro...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 20.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355064 (CHEMBL1834616) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360418 (CHEMBL1934264) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244437 ((2R,3S)-4-(4-tert-butylphenylsulfonyl)-2,3-dihydro...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25.3 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360416 (CHEMBL1934260) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355059 (CHEMBL1834620) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 31.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244619 ((2R,3S)-4-(3-chlorophenylsulfonyl)-2,3-dihydroxy-N...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 85.9 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360419 (CHEMBL1934253) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360421 (CHEMBL1934259) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 122 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360417 (CHEMBL1934265) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 139 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244439 ((2R,3S)-4-(2,3-dichlorophenylsulfonyl)-2,3-dihydro...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 141 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360424 (CHEMBL1934255) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >160 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50244618 ((2R,3S)-2,3-dihydroxy-N-((R)-6-(piperidin-1-ylmeth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assay | Bioorg Med Chem Lett 18: 4764-9 (2008) Article DOI: 10.1016/j.bmcl.2008.07.108 BindingDB Entry DOI: 10.7270/Q29C6X87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360420 (CHEMBL1934254) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 248 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355070 (CHEMBL1834749) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 342 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Inhibition of rabbit B1 receptor by cellular calcium flux assay | J Med Chem 54: 7232-46 (2011) Article DOI: 10.1021/jm200808v BindingDB Entry DOI: 10.7270/Q28C9WP1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360422 (CHEMBL1934256) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 393 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50209720 ((R)-3-(4-fluorophenyl)-N-((R)-7-(pyrrolidin-1-ylme...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 451 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor | J Med Chem 50: 2200-12 (2007) Article DOI: 10.1021/jm070055c BindingDB Entry DOI: 10.7270/Q2MS3SG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355069 (CHEMBL1835756) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 476 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360414 (CHEMBL1934262) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >800 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360423 (CHEMBL1934258) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >800 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360425 (CHEMBL1934257) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >800 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50209726 ((R)-3-(4-fluorophenyl)-N-((R)-7-((2-methoxyethylam...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit bradykinin B1 receptor | J Med Chem 50: 2200-12 (2007) Article DOI: 10.1021/jm070055c BindingDB Entry DOI: 10.7270/Q2MS3SG2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360413 (CHEMBL1934261) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50360415 (CHEMBL1934263) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B1 bradykinin receptor (Oryctolagus cuniculus) | BDBM50355083 (CHEMBL1835762) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >6.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc. Curated by ChEMBL | Assay Description Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cells | Bioorg Med Chem Lett 22: 619-22 (2011) Article DOI: 10.1016/j.bmcl.2011.10.068 BindingDB Entry DOI: 10.7270/Q25X29CW | |||||||||||
More data for this Ligand-Target Pair |